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N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-(2-methyl-2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]propanamide
2-{2-[3-(2-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-2-azaspiro[4.4]nonan-3-one
N-benzyl-N-methyl-3-({methyl[4-(morpholin-4-yl)butyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-(5-acetylthiophen-3-yl)-N-[(3S)-1-benzylpyrrolidin-3-yl]acetamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-propyl-1H-pyrazole-5-carboxamide
(3S,4S)-1-(benzenesulfonyl)-4-[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]pyrrolidin-3-ol
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-3-(piperidin-3-yl)benzamide
4-methoxy-N-methyl-3-(3-methyl-1H-pyrazol-1-yl)benzamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-2-yl)ethyl]amine
7-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2,3-dimethyl-1H-indole
3-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)-N-(1,3-thiazol-2-ylmethyl)propanamide
(1S,5R)-6-(1-ethyl-1H-pyrazole-5-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-(2-{[4-(trifluoromethyl)pyridin-2-yl]oxy}hex-5-en-1-yl)morpholine
1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-4-(6-methylpyridin-2-yl)piperazine
2-cyclopropyl-6-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,6-dihydropyrimidine-5-carboxamide
N-{3-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-oxopropyl}methanesulfonamide
1-[1'-(2-fluoro-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
5-cyclopropanecarbonyl-1'-(quinolin-6-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-(5-methyl-1,3,4-oxadiazol-2-yl)-6-(morpholin-4-yl)-decahydroisoquinoline
3-(2,3-difluorobenzoyl)-9-methoxy-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-amino-1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-N-(2-methylpropyl)-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
5-[(3-hydroxypiperidin-1-yl)methyl]-N-{[4-(trifluoromethoxy)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]methanesulfonamide
3-(3-chlorobenzoyl)-1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperidine
N-methyl-N-(1,2-oxazol-3-ylmethyl)-3-[(3S,4R)-1-(propan-2-yl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
4-(1-benzyl-1H-pyrazole-4-carbonyl)-1-(4-methylphenyl)piperazin-2-one
1-{2-[1-(2-phenylethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]piperidin-1-yl}ethan-1-one
4-(3-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)-2-methylbutan-2-ol
1-[2-(benzyloxy)ethyl]-3-ethylpiperidine-3-carboxylic acid
4-(1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-4-yl)pyridine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(1R,5S,6R)-3-{[2-(trifluoromethyl)phenyl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
5-{[benzyl(methyl)amino]methyl}-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1,2-oxazole-3-carboxamide
N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-ethyl-1'-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
N-{2-[1-(2,4-dichlorobenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-3-(2-oxopyrrolidin-1-yl)propanamide
methyl 4-{4-[2-(thiophen-3-yl)acetyl]piperazin-1-yl}benzoate
1-(2-methylphenyl)-4-(2-phenoxypropanoyl)piperazin-2-one
[1-({4-[(2H-1,3-benzodioxol-5-yl)amino]-8-methylquinazolin-2-yl}methyl)piperidin-4-yl](thiophen-2-yl)methanol
1-[cyclohexyl(methyl)amino]-3-(3-{[cyclopropyl(ethyl)amino]methyl}phenoxy)propan-2-ol
4-(2,6-dimethylpyridin-3-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-2-amine