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N-(1-hydroxybutan-2-yl)-N-[(2-methylphenyl)methyl]-3-(2-oxopiperidin-1-yl)propanamide
(3R,5S)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(2-phenylethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-3-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(piperidin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(2,5-dimethoxybenzoyl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-9H-purine
(4aS,8aR)-2-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)-decahydroisoquinoline
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)-2-(1H-pyrazol-1-yl)acetamide
5-(2,4-difluorophenoxymethyl)-N-(1-hydroxy-2-methylpropan-2-yl)-1,2-oxazole-3-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
3-(1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[2-(pyridin-2-yl)ethyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}azocane
2-ethyl-9-(2-methyl-1,3-thiazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
1-methyl-2-oxo-8-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(cyclohex-1-en-1-ylmethyl)-3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
1-(cyclopropylmethyl)-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]carbamoyl}-2,1,3-benzoxadiazol-1-ium-1-olate
4-{[3-(difluoromethoxy)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
2-{[5-(pyridin-3-yl)-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-1,4-oxazepan-6-yl}methanol
methyl 1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-4-carboxylate
1-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-3-ethylpiperidine-3-carboxylic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(quinoxalin-2-yl)piperidin-3-ol
4-hydroxy-1-[4-(1H-pyrazol-4-yl)butanoyl]piperidine-4-carboxylic acid
N-[4-(3,5-dimethoxyphenyl)phenyl]-2-methoxyacetamide
4-(3-methylbutyl)-11-{[2-(pyridin-2-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4,5-dimethyl-2-{3-[4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]propyl}-1H-1,3-benzodiazole
2-(4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-1-yl)pyridine-3-carbonitrile
3-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrrolidin-3-yl)methyl]benzoic acid
2,6-dimethyl-4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
2-(3-phenylpropyl)-8-(pyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}thiomorpholine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
3-(2H-1,3-benzodioxol-5-yl)-5-(1-phenoxypropan-2-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-methyl-5-(2-phenylphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-[1-(3-ethynylbenzoyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-1-{4-[2-(4-methylphenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
3-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)-3-propylurea
N-benzyl-1-{imidazo[1,2-a]pyridine-2-carbonyl}-N-methylpiperidin-3-amine
(4aR,7aS)-1-(2-methoxyethyl)-4-[(3-methyl-1-benzofuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(methoxymethyl)cyclopentyl]-3-azaspiro[5.5]undecan-9-amine
ethyl 4-[1-(2-methylpropyl)-2,4-dioxo-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
4-({2-[1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-{1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
2-[9-(2-hydroxy-4-methoxybenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetic acid
5-{[benzyl(methyl)amino]methyl}-N-(3-hydroxy-2,2-dimethylpropyl)-N-methyl-1,2-oxazole-3-carboxamide