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5-{2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}methyl)phenyl]ethan-1-one
8-[6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-[(1R,5R)-6-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-(3-{4-[(2-phenylpropyl)amino]piperidin-1-yl}phenyl)cyclopropanecarboxamide
5-ethyl-N-({3-methyl-7-[4-(thiophen-2-yl)butanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,2-oxazole-3-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
2-[(2-chlorophenyl)methyl]-4-[(trimethylpyrazin-2-yl)methyl]morpholine
N-[(3S,4R)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-(5-ethyl-2-methylpyrimidin-4-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
1-(4-{[1-(dimethylamino)butan-2-yl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(4aS,8aR)-6-({8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
3-(5-methyl-2-oxo-5-phenylpiperidin-1-yl)propanoic acid
(3R)-1-(5-fluoro-2-methoxybenzoyl)-3,4,4-trimethylpyrrolidin-3-ol
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-(2-methanesulfonylethyl)acetamide
1-benzyl-4-[1-(2-methoxyacetyl)piperidine-4-carbonyl]piperazin-2-one
{4-[({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)methyl]oxan-4-yl}methanol
4-chloro-3-[1-(1-methanesulfonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1-methyl-1H-indazole
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-[methyl(piperidin-4-yl)amino]acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-6-methyl-N-(oxolan-2-ylmethyl)pyridine-2-carboxamide
N,2-dimethyl-N-(2-phenyl-1-{1-[(2E)-3-phenylprop-2-enoyl]piperidin-4-yl}ethyl)furan-3-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[(4-acetamidophenyl)methyl]piperidin-3-yl}propanamide
7-(naphthalene-1-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(2-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
1-{2-[cyclopentyl(methyl)amino]ethyl}-3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-5-yl}-1-methylurea
5-cyclopropanecarbonyl-1'-(1-methyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{[4-(2,4-dimethylphenyl)piperazin-1-yl]methyl}-4-(pyrazin-2-yl)phenol
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-5-propyl-1,2-oxazole-3-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(1H-imidazol-4-ylmethyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-methylpyrido[2,3-d]pyrimidin-4-amine
(2S)-1-({4-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]phenyl}methyl)pyrrolidine-2-carboxylic acid
4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(thiophen-3-ylmethyl)piperidine
4-({1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
6-[(diethylamino)methyl]-N-(3-hydroxypropyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl[(4-methyl-1,3-thiazol-2-yl)methyl](2-phenoxyethyl)amine
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-fluoro-6-methoxybenzamide
(1-{1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}ethyl)dimethylamine
N-(2-methoxyethyl)-1-{1-[3-(4-methylphenyl)propanoyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
methyl 1-[(3R,5S)-1-cyclopentyl-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{2-[2-(propan-2-yloxy)phenyl]ethyl}thiolan-3-amine
1-(2-chlorophenyl)-4-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-1H-indole-6-carboxamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-[methyl(phenyl)amino]ethan-1-one
1-(benzenesulfonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(1R,5R)-N,N-dimethyl-6-(5-propylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-hydroxybutanamide