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(4aS,8aR)-1-(3-aminopropyl)-6-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
4-[1-(1-methylpiperidin-4-yl)-4-phenyl-1H-imidazol-5-yl]benzoic acid
2-chloro-N-[2-({2-[(dimethylamino)methyl]-1,3-thiazol-4-yl}formamido)ethyl]benzamide
2-(4-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)ethan-1-ol
N-(1-cycloheptylpiperidin-3-yl)-5-methyl-1,3-oxazole-4-carboxamide
1-cyclohexyl-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
5-methyl-3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N-({5-[(2-fluoro-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
1-[(2-fluorophenyl)methyl]-N-{2-[2-(trifluoromethyl)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
3-{[4-(6-ethoxy-4-methylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}phenol
5-(2-{3-cyclohexyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(3-hydroxypropyl)amino]pyridine-3-carboxamide
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
1-[2-(4-chlorophenyl)ethyl]-5-[4-(2-hydroxyethyl)piperazine-1-carbonyl]piperidin-2-one
(2S)-2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-3-(1H-indol-3-yl)propan-1-ol
(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-1,2,3,6-tetrahydropyridine
2-(dimethylamino)-2-(4-fluorophenyl)-N-(1,2-oxazol-3-ylmethyl)acetamide
(3aS,6aS)-2-cyclopentyl-5-[(2,5-dimethylphenyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 1-[(3S,5S)-5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]carbamoyl}-1-{[5-(2-chlorophenyl)furan-2-yl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[1-(pyridin-4-yl)propyl]-1,3-oxazole-4-carboxamide
8-(5-ethyl-1,2-oxazole-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
6-{3-methylimidazo[1,5-a]pyridin-1-yl}-5-phenyl-1H-pyrazolo[3,4-b]pyridine
5-fluoro-2-methyl-3-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
2-ethyl-8-(2-ethylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
6-[(2R)-1-hydroxy-3-methylbutan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-methyl-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-methyl-1-benzofuran-5-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(1H-indazol-1-yl)acetamide
3-[4-(1-methoxyethyl)phenyl]-6-(propan-2-yloxy)pyridazine
2-({4-[4-(hydroxymethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
3-(methanesulfonylmethyl)-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidine
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methylacetamide
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
1-[(5-methylfuran-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
N-(4-aminobutyl)-3-[(4-fluorophenyl)formamido]propanamide
2-amino-8-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-benzyl-6-[3-(morpholin-4-ylmethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-[(2-fluoro-5-methoxyphenyl)methyl]pyrrolidin-2-one
1'-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(oxan-4-yl)-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-(1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-phenylethyl)-N-methylpyridine-2-carboxamide
2-(6-chloropyridin-3-yl)-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
2-({[(6-hydroxy-1,4-oxazepan-6-yl)methyl](methyl)amino}methyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-[(6-methoxypyrimidin-4-yl)amino]-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine