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2-(4-methyl-1H-pyrazol-1-yl)-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-yl)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-3-amine
2-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-amine
1-(2-hydroxyethyl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1H-1,3-benzodiazole-5-carboxamide
1-(4,6-dimethylpyrimidin-2-yl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
(1S,5R)-3-[(1-phenyl-1H-pyrazol-4-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(5S,9aS,9bS)-5-(2-fluoro-4-methoxyphenyl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]-3-(4-fluorophenyl)propanoic acid
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2,6-dimethylpyridine-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}acetamide
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-{2-[1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]ethyl}acetamide
3-[(1,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(isoquinolin-1-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]amine
(4aR,7aS)-1-acetyl-4-[(4-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-acetyl-N-(1-{2-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
5-methoxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,3-dimethyl-1H-indole-2-carboxamide
8-(2,6-dimethoxypyridine-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[(4aR,7aS)-4-[2-(4-methoxyphenyl)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-(2-methoxyphenyl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(2-methoxypyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-(furan-2-ylmethyl)piperidine
2-(4-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}morpholin-3-yl)acetic acid
(2S,4S)-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)-4-[(pyridin-4-ylmethyl)amino]pyrrolidine-2-carboxamide
[(3R,5R)-1-(5,6-dimethylpyridine-3-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
3-({1-[3-(2-methylphenyl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
ethyl 4-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine-1-carboxylate
(2R)-2-hydroxy-2-phenyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
3-{4-[6-amino-5-cyano-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}propanoic acid
(4S)-4-hydroxy-3,3,4-trimethyl-N-[(2-methylphenyl)methyl]piperidine-1-carboxamide
N-(5-oxo-1-propylpyrrolidin-3-yl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
4-{[3-(2-methoxyethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
methyl 5-(benzylamino)-3-(4-methoxybenzamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-hydroxy-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-3-ol
N-(cyclobutylmethyl)-N-(oxolan-2-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(1,3,4-thiadiazol-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[1-(3,5-dimethylphenyl)-1H-imidazol-2-yl]-N,N-dimethylpyrimidin-2-amine
4-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
1-(2,6-dimethylpyridin-4-yl)-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
2-[2-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(1,2,5-oxadiazole-3-carbonyl)-1,4-diazepan-6-ol
N-[(1S)-1-[1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propyl]acetamide