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2-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-N-methylacetamide
4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1λ6-thiane-1,1-dione
(1R,3S)-3-(2-aminoethoxy)-7-[(3-chloro-4-methoxyphenyl)methyl]-7-azaspiro[3.5]nonan-1-ol
3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
8-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-ethyl-2-{4-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]morpholin-3-yl}acetamide
N-cyclopropyl-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(2S)-3-phenyl-2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propanamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-3-(1H-indol-3-yl)propanamide
2-[(1S,5R)-6-[(4-methoxy-2,5-dimethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
4-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1-(2-methoxyethyl)pyrrolidin-2-one
dimethyl({4-methyl-5-[1-(piperidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
2-(2-hydroxyphenyl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
1-(4-methylphenyl)-4-[4-(morpholin-4-yl)pentanoyl]piperazin-2-one
N-(2-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-{5-cyclopropyl-4-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2-fluorophenyl)pyrimidine
N-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]-4-(pyridin-3-yloxy)piperidine-1-carboxamide
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-3-ol
4-(cyclopropylsulfamoyl)-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
3-(2H-1,3-benzodioxol-5-yl)-N-(carbamoylmethyl)-3-phenylpropanamide
N-[2-(3-methoxyphenyl)ethyl]-6-[2-(thiophen-2-yl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(1-ethylpiperidin-3-yl)-1H-1,3-benzodiazole-6-carboxylic acid
1-(1-ethylpyrrolidine-2-carbonyl)-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
9-[2-(4-fluorophenyl)acetyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-3-cyclobutyl-4-methyl-1-[4-(pyrrolidin-1-ylmethyl)benzoyl]pyrrolidin-3-ol
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-4-propylpyrimidine-5-carboxamide
2-[methyl({[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]-N-(1,3-thiazol-2-yl)propanamide
1-methyl-3-(pyridin-3-yl)-4-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
6-chloro-3-({[(4-ethylphenyl)methyl](methyl)amino}methyl)-N,N-dimethylimidazo[1,2-a]pyridine-2-carboxamide
1-ethyl-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-N-[2-(pyridin-2-yl)ethyl]-1-(pyridin-3-ylmethyl)piperidin-3-amine
butyl 8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-methoxypropan-1-one
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[(3-methylpyridin-4-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
6-methyl-5-{2-oxo-2-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridin-4-amine
8-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-methoxyethyl)-9-[2-(2-methoxyphenoxy)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-cycloheptylpiperidin-3-yl)-3-[4-(dimethylamino)phenyl]propanamide
N-(furan-2-ylmethyl)-N,1-dimethyl-5-[methyl(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2-methoxyethyl)-4-[1-(2-methoxyphenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
3-[2-(1-cyclopentylpiperidin-2-yl)ethyl]-6-methyl-3,4-dihydroquinazolin-4-one
1-(dimethylamino)-3-(4-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-[2-(dimethylamino)ethyl]-N-[2-(4-methylphenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-[1-({1-[(5-ethylthiophen-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea