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(4aR,7aS)-1-(cyclopropylmethyl)-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1S,2S)-2-hydroxycyclohexyl]-5-{[methyl(2-phenylethyl)amino]methyl}-1,2-oxazole-3-carboxamide
4-[5-(2,3-dihydro-1H-inden-2-yl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]morpholine-2-carboxamide
N-[1-(morpholin-4-ylmethyl)cyclopentyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
3-[(3R,4S)-4-(dimethylamino)-1-[2-(4-fluoro-2-methylphenyl)acetyl]piperidin-3-yl]propanoic acid
(2R,3R,6R)-5-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}benzoic acid
5-phenyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
2-{2-[1-cyclohexyl-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
(3aR,6aR)-2-methanesulfonyl-5-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(3R,4R)-3-hydroxy-1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-4-yl]pyridine-4-carboxamide
1-(2-chloro-4-fluoro-5-methylphenyl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
N-(2-methoxyethyl)-2-methyl-7-{[(1s,4s)-4-aminocyclohexyl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[5-({[2-(2-ethyl-1H-imidazol-1-yl)ethyl]carbamoyl}amino)-2-fluorophenyl]-2-methylpropanamide
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-2,3-dihydro-1-benzofuran-5-carboxamide
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
3-[2-(1H-imidazol-1-yl)acetyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
5-(4-acetylphenoxymethyl)-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2-oxazole-3-carboxamide
N-({7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methylbutanamide
(4aS,7aR)-1-[2-(furan-2-yl)-2-oxoacetyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-methyl-4-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
3-butanamido-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methylbenzamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-tert-butyl-1-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]urea
N-{[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzenesulfonamide
N-[1-(4-methylphenyl)ethyl]-2-({[6-(trifluoromethyl)pyridin-3-yl]methyl}amino)acetamide
N-({1-[(2-hydroxy-7-methylquinolin-3-yl)methyl]pyrrolidin-3-yl}methyl)-2-methoxyacetamide
3-[2-(piperidin-1-yl)ethyl]-1-[4-(pyridin-2-ylmethoxy)phenyl]urea
2-methoxy-4-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]pyridine-3-carbonitrile
(2S,4R)-N,N-diethyl-1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
methyl N-[(3S,5S)-5-{[(2-fluorophenyl)methyl]carbamoyl}-1-methylpyrrolidin-3-yl]carbamate
(3S,4R)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1-benzothiophene-2-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(morpholin-4-yl)ethyl]amine
2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-5-methoxyphenol
7-hydroxy-6-methyl-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,3,4-tetrahydroquinolin-2-one
3-({[(4,6-dimethylpyrimidin-2-yl)methyl]amino}methyl)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-(3-chloro-4-hydroxyphenyl)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
5-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-(2-methylpropyl)-1H-imidazole
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
3-amino-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]pyrrolidine-3-carboxylic acid
6-chloro-N,N-dimethyl-3-[({[4-(morpholin-4-yl)phenyl]methyl}amino)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-[4-(benzyloxy)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
2-(benzyloxy)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
ethyl 3-({5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}amino)propanoate
2-amino-4-(3-hydroxy-4-methoxyphenyl)-6-(4-methylthiophen-2-yl)pyridine-3-carbonitrile
N-benzyl-N-methyl-3-(quinolin-5-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide