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2-amino-3-ethyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
1-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-4-phenylpiperazine
2-chloro-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-(piperidine-1-carbonyl)aniline
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pyrazine-2-carboxamide
7-methyl-2-(4-phenoxybutanoyl)-2,7-diazaspiro[4.5]decan-6-one
2-(dimethylamino)-2-(3-methylphenyl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}acetamide
1-{1-[2-(methylamino)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
1-(oxan-4-yl)-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
4-({3-[4-(1H-imidazol-1-ylmethyl)phenyl]phenyl}methyl)morpholine
N,N-dimethyl-3-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}aniline
7-(2-hydroxyethyl)-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
N,2-dimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1,3-benzoxazole-6-carboxamide
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-[2-(4-methoxyphenyl)ethyl]-2-methyl-N-[(1-methylpiperidin-4-yl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2,2,6,6-tetramethyl-N-(4-phenylbutan-2-yl)piperidin-4-amine
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-4-carboxamide
5-(methanesulfonylmethyl)-2-(4-methanesulfonylphenyl)pyridine
2-{4-[4-(2-fluorophenoxy)piperidine-1-carbonyl]piperidin-1-yl}-4-methyl-6-(propan-2-yl)quinazoline
1-[4-methyl-6-(methylamino)pyrimidin-2-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-[1-({1-[1-(4-fluorophenyl)pyrrolidin-3-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-ol
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-2-hydroxy-2-(4-methoxyphenyl)ethan-1-one
7-methyl-2-(6-methyl-2-propylpyrimidin-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(1-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
4-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]pyrimidin-2-amine
2-amino-6-(4-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)pyrimidin-4-ol
9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-3-[(2,3,6-trifluorophenyl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(propan-2-yl)acetamide
(1-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
3-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-1-[(1r,4r)-4-hydroxycyclohexyl]urea
2-amino-4-[2-(ethylamino)pyrimidin-5-yl]-6-(3-methylphenyl)pyridine-3-carbonitrile
4-ethyl-1-(2-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-2-oxoethyl)-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[1-(2-phenoxyethyl)piperidin-3-yl]-1H-1,3-benzodiazole
1-(2-methoxyphenyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
(2S,4R)-1-methyl-N-(propan-2-yl)-4-{2-[2-(trifluoromethyl)phenyl]acetamido}pyrrolidine-2-carboxamide
N3-(cyclopropylmethyl)-N5-[(4-methylphenyl)methyl]-4-oxo-N3-propyl-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[2-({[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}(methyl)amino)ethyl]cyclopentan-1-ol
N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,3-oxazole-4-carboxamide
[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
4-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
2-(morpholin-3-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]acetamide
(1S,5R)-6-benzyl-3-[(5-methylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-cyclopentyl-N-[(2-methoxyphenyl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(1R,3S)-7-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-7-azaspiro[3.5]nonane-1,3-diol
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylpropanamide
3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-5,6,7,8-tetrahydroquinoline
8-methoxy-2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}quinoline