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1-(2-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-4-methylpyrimidin-5-yl)ethan-1-one
6-[3-(pyridin-3-yl)azetidin-1-yl]pyridine-2-carbonitrile
9-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-{5-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)methyl]-1-methyl-1H-pyrrol-3-yl}ethan-1-one
3-(3-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-ylmethyl}-1H-indol-1-yl)propanamide
6-(benzyloxy)-1-cyclohexyl-4-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-1,4-diazepan-2-one
(1R,5R)-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-5-(trifluoromethyl)pyridine
1-(1-methyl-1H-pyrazole-3-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-(2-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
1-(4-methylquinazolin-2-yl)-N-[(1S)-1-phenylethyl]pyrrolidine-2-carboxamide
(1-{5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carbonyl}piperidin-3-yl)methanol
1-benzyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-1H-pyrazole-4-carboxamide
2-methyl-4-(5-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}furan-2-yl)but-3-yn-2-ol
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
butyl(furan-2-ylmethyl){[2-(morpholin-4-yl)pyridin-3-yl]methyl}amine
1-{[(3R,4R)-1-[(3,4-dimethylphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
2-methyl-4-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]quinoline
N-{[7-(2-methoxy-2-phenylacetyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-methylthiophene-2-carboxamide
[4-benzyl-1-(3,4-dimethoxybenzenesulfonyl)piperidin-4-yl]methanol
5-(methoxymethyl)-N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-2-carboxamide
2-cyclopentyl-1-{4-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}ethan-1-one
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
methyl({[2-(propan-2-yl)pyrimidin-5-yl]methyl})[2-(pyridin-4-yl)ethyl]amine
2-(dimethyl-1,2-oxazol-4-yl)-1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
N-(2-hydroxyethyl)-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(propan-2-yl)acetamide
(3S,4S)-4-(dimethylamino)-1-[(3-fluoro-2-methoxyphenyl)methyl]pyrrolidin-3-ol
methyl(3-methylbut-2-en-1-yl)({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
{5-[1-(2-methylphenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]furan-2-yl}methanol
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
[(3,4-difluorophenyl)methyl](methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
1-{[3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazin-1-yl]methyl}naphthalen-2-ol
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethylpent-4-ynamide
2-(2,3-dimethoxyphenyl)-4-(trifluoromethyl)pyridine
1-[(2-chlorophenyl)methyl]-7-(methylsulfanyl)-3-(morpholin-4-ylmethyl)-1,2-dihydroquinolin-2-one
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}-1-(furan-3-ylmethyl)piperidine
1-(2-hydroxyethyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}piperidine-4-carboxamide
2-amino-3-ethyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}pentane-1,5-diamine
N-{2-[({1-[(3,4-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]ethyl}acetamide
2-[4-(6-ethyl-2-methylquinoline-4-carbonyl)-1-methylpiperazin-2-yl]ethan-1-ol
1-{3-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]phenyl}ethan-1-one
3-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-4-yl}-N-cyclopropylpropanamide
3-methyl-1-(2-methylpropyl)-8-[(2,4,6-trimethoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-oxoethyl}-2-methyl-1,4-dihydroquinolin-4-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
(3R,4S)-4-(5-methylfuran-2-yl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-amine
6-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]pyridine-2-carbonitrile
N-[(5-methyl-1H-pyrazol-3-yl)methyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide