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N-ethyl-N-(2-methylprop-2-en-1-yl)-7-oxo-2-(thiophene-3-amido)-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
(3R,4R)-3-methyl-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]-4-(oxan-4-yl)piperidin-4-ol
3-(5-methanesulfonamido-2-methylphenyl)-1-[3-(morpholin-4-yl)propyl]urea
5-methoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-indole-2-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
2-{[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]methyl}benzonitrile
N-methyl-N-({5-[(2-methyl-5-oxo-1,4-diazepan-1-yl)methyl]furan-2-yl}methyl)methanesulfonamide
N-cyclopropyl-3-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}propanamide
N,N-dimethyl-4-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]benzamide
N-benzyl-2-(2-methoxyphenyl)pyrrolidine-1-sulfonamide
2-(1H-pyrazol-1-yl)-1-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)butan-1-one
1-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}azepane-2-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-ethyl-N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
2-[(2-chlorophenyl)methyl]-4-{4-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-(1-{1-[4-(4-methoxyphenyl)-4-oxobutanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-3-(thiophen-2-yl)-1H-pyrazol-4-yl)methanol
5-{[methyl({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}pyrimidin-2-amine
(1S,5R)-N,N-diethyl-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-sulfonamide
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)butane-1-sulfonamide
ethyl 3-{[3-(dimethylcarbamoyl)-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
butyl({[2-(ethylsulfanyl)pyrimidin-5-yl]methyl})(furan-2-ylmethyl)amine
4-(cyclopropylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-5-one
3-chloro-N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-6-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
(1S,6R)-9-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{1-[5-(hydroxymethyl)furan-2-carbonyl]pyrrolidin-3-yl}propan-2-ol
N-methyl-3-(morpholine-4-carbonyl)-N-(oxan-4-yl)benzene-1-sulfonamide
2-butyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-2,5-dihydro-1H-pyrrole
3-(3,4-dimethoxybenzoyl)-1-phenylmethanesulfonylpiperidine
N,N-dimethyl-5-(1-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1H-imidazol-2-yl)pyrimidin-2-amine
1-{[(4-fluorophenyl)methyl]carbamoyl}-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-cyclopropyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-4-(pyridin-2-yl)pyrimidine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-benzylpyrrolidin-3-amine
N-(1H-1,3-benzodiazol-2-ylmethyl)-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
(5S)-5-{[benzyl({[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl})amino]methyl}pyrrolidin-2-one
5-cyclopropyl-N-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-oxo-2-phenyl-N-(pyridin-3-ylmethyl)acetamide
N3-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-(2-{7-[(2-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
N-{[7-(2,5-difluorobenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-4-carboxamide
8-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]isoquinoline
N-[4-(1H-pyrazol-4-yl)phenyl]-2-(pyrrolidin-3-yl)benzamide
2-{4-[(3-ethoxyphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-[2-(dimethylamino)ethyl]-2-(2-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-[(3S,4R)-1-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-{2-[2-(3-fluorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide