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N-[2-(2-methyl-1H-indol-3-yl)ethyl]-3-(2-oxoazepan-1-yl)propanamide
4-(5-{[2-(difluoromethoxy)phenyl]methyl}-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)morpholine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole
3-{2-[4-(2,3-dimethylphenyl)piperazin-1-yl]-2-oxoethyl}-4-[(2-fluorophenyl)methyl]piperazin-2-one
2-(4-{4-[ethyl(methyl)amino]pyrimidin-2-yl}-1H-pyrazol-1-yl)-N-(1-methyl-1H-indazol-3-yl)acetamide
(2S,4S)-1-benzyl-4-{[(3-chlorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[4-(trifluoromethyl)phenyl]ethyl}propanamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-propylpiperidin-4-yl)acetamide
5-methyl-N-{[1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-3-yl]methyl}-1,2-oxazole-3-carboxamide
1-methyl-5-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)furan-2-carboxamide
(1S,5R)-6-(2,6-difluoro-3-methoxybenzoyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)pyridine-2-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(morpholin-3-yl)acetamide
1-ethyl-3-(oxan-4-yl)-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
2-(3-methylbutyl)-8-{spiro[2.4]heptane-1-carbonyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-[2-(ethylamino)pyrimidin-5-yl]-1-(4-methoxyphenyl)-3-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxybutan-1-one
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(quinoxalin-6-ylmethyl)acetamide
3-{[1-(3-hydroxypyridine-2-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-benzyl-N-(2-hydroxyethyl)-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
5-fluoro-N2,N4,N4-trimethyl-N2-[(2-methylpyridin-4-yl)methyl]pyrimidine-2,4-diamine
N-{2-[1-(2-acetamidoethyl)-1,2,3,6-tetrahydropyridin-4-yl]ethyl}piperidine-1-carboxamide
2-[(2-fluorophenyl)methyl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1,3-benzoxazole-6-carboxamide
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(4-fluorophenyl)morpholine
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N,4-dimethylpyrimidin-2-amine
2-ethyl-4-{1-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
2-{4-[2-(3-methoxyphenoxy)ethyl]phenyl}-1,3,4-oxadiazole
N-[(3R,4S)-1-(2-cyclopentylacetyl)-4-phenylpyrrolidin-3-yl]methanesulfonamide
3-methyl-7-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{1-azabicyclo[2.2.2]octan-3-yl}-4-(3-hydroxy-3-methylbutyl)benzamide
(4-{[2-(methylsulfanyl)phenyl]methyl}morpholin-3-yl)methanol
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-cyclopentyl-1,4-diazepane
1-({3-cyclopropyl-1-[2-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}methyl)-1,2-dihydropyrimidin-2-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(3-methoxypropyl)acetamide
N-(2-{7-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
methyl 4-[ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})carbamoyl]butanoate
methyl (2S,4S)-4-(2-methoxypyrimidine-5-amido)-1-methylpyrrolidine-2-carboxylate
7-(azepan-1-ylmethyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-indole-3-carboxamide
6-cyclopentyl-1-methyl-4-{3-methyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}-1H-pyrazolo[3,4-d]pyrimidine
N-{[(1R,2R)-2-hydroxycyclohexyl]methyl}-4-(quinolin-5-yloxy)piperidine-4-carboxamide
3-{[3-cyclopropyl-1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}phenol
1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-N-[1-(thiophen-2-yl)propan-2-yl]piperidine-4-carboxamide