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9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-{[5-(1-benzylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}-4-methylpiperazine
2-{methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
1-[(2-fluorophenyl)methyl]-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-1-[(2,6-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(2-methyl-1,3-benzothiazol-5-yl)pyrrolidine-2-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-methyl-N-(oxan-4-yl)pyridin-2-amine
1-(4-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}phenyl)-1H-1,2,4-triazole
3,4-dimethoxy-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-[(5-methoxy-1H-indol-2-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
5-methoxy-2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
3-[3-(2-methoxyethyl)-1-(4-methylphenyl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroisoquinolin-1-one
4-chloro-2-({4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
2-(5-{5-butyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}furan-2-yl)benzonitrile
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
5-(2-methyl-1H-imidazole-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(pyrimidin-2-yl)-1,4-diazepane
(4-{[5-(oxan-2-yl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
5-(furan-3-ylmethyl)-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)cyclohexanecarboxamide
1,3-dimethyl-N-(oxan-4-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[2-(benzyloxy)ethyl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
4-(2,3-dimethyl-1H-indole-7-carbonyl)-7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-N-(propan-2-yl)piperidine-1-carboxamide
2-methyl-7-oxo-N-{1-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
2-amino-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-(2-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
4-{1-[(4-chlorophenyl)methyl]-6-oxopiperidine-3-carbonyl}-1-phenylpiperazin-2-one
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidin-3-yl)piperazine
N-[(2-methoxyphenyl)methyl]-2-methyl-N-(prop-2-en-1-yl)furan-3-carboxamide
5-chloro-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)thiophene-2-sulfonamide
N-[7-(azocane-1-carbonyl)-1-ethyl-2-(3-methoxyphenyl)-1H-1,3-benzodiazol-5-yl]acetamide
4-[(2-hydroxyethyl)sulfanyl]-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]benzamide
4-[1-(piperidin-4-yl)piperidine-3-carbonyl]morpholine
N-[(3R,4S)-4-cyclopropyl-1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]pyrrolidin-3-yl]methanesulfonamide
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3-phenoxypropanamide
2-ethoxy-3-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyridine
(2S,4S)-4-amino-1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
1-(4-benzylpiperazin-1-yl)-3-{1-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]piperidin-3-yl}propan-1-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-(1-methyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[4-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperazin-1-yl]phenol
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-(2-{4-[(2-ethylbutanamido)methyl]-5-methyl-1,3-oxazol-2-yl}phenyl)oxolane-2-carboxamide
1-{[3-(benzyloxy)phenyl]methyl}azepan-4-ol
2-(5-acetylthiophen-3-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
methyl (2S,3S)-2-{[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]formamido}-3-methylpentanoate
1-[(5-methylfuran-2-yl)methyl]-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid