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3-(3-methoxyphenyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]-1H-pyrazole-5-carboxamide
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
1-(6-methoxypyridin-2-yl)-5-methyl-1H-pyrazole-3-carboxylic acid
methyl 4-{[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}butanoate
6-methyl-2-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2-dihydroquinoline-4-carboxamide
N-[2-(1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazol-4-yl)ethyl]acetamide
1-(2-ethoxypyridine-3-carbonyl)-4-(furan-2-carbonyl)-1,4-diazepane
(1R,3S)-7-(4-methanesulfonylbenzoyl)-7-azaspiro[3.5]nonane-1,3-diol
N-[3-(3-methylpyrazin-2-yl)phenyl]acetamide
4-{[4-(5-ethylpyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-N,N-dimethylaniline
N,N-dimethyl-N'-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanediamide
5-tert-butyl-4-({5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)furan-2-carboxamide
3-[(benzylamino)methyl]-1-[(2,3-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
3-(2,6-dimethoxypyridin-3-yl)-1-(oxolan-2-ylmethyl)-1-(pyridin-2-ylmethyl)urea
2-{4-[(3,5-dimethoxyphenyl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-methyl-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]-1-(oxan-4-yl)piperidine
5-{3-[4-(2-ethoxyphenyl)piperazin-1-yl]-3-oxopropyl}-5-[(4-methoxyphenyl)methyl]pyrrolidin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-methylbenzamide
3-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole
2-[(1-ethylpyrrolidin-2-yl)methyl]-N-[(5-methylfuran-2-yl)methyl]-3-oxo-2,3-dihydro-1H-isoindole-5-carboxamide
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-2-phenoxyethan-1-one
methyl 1-({2-[benzyl(methyl)carbamoyl]imidazo[1,2-a]pyridin-3-yl}methyl)piperidine-2-carboxylate
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-hydroxypropan-1-one
4-(4-chlorophenoxy)-N-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidine-4-carboxamide
1-(methoxymethyl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)cyclobutane-1-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
4-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-6-(morpholin-4-yl)pyrimidin-2-amine
1-ethyl-8-[(2-hydroxy-3-methoxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propyl]piperidine-3-carboxamide
N-{2-[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}cyclohexanecarboxamide
N-[1-methyl-3-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)-1H-pyrazol-5-yl]acetamide
N-{[1-(6-cyanopyridine-3-carbonyl)piperidin-3-yl]methyl}-1H-indazole-3-carboxamide
2-(4-{[(quinolin-7-yl)amino]methyl}phenoxy)ethan-1-ol
(2S,4S)-4-[(cyclohexylmethyl)amino]-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
2-(4-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
2-{1-benzyl-4-[(2,4,5-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(2-methoxyphenoxy)ethan-1-one
(3E)-1-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pent-3-en-1-one
2-amino-4-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
1-{2-methyl-4-[3-(2-methylphenyl)piperidin-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-1H-indole-3-carbonitrile
methyl({[5-(1H-pyrazol-3-yl)furan-2-yl]methyl})(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
ethyl 5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
9-methoxy-3-methyl-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
methyl 4-{5-chloro-2-[(2-acetamido-3-methylbutanamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}benzoate
3-[3-(oxan-4-yl)-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
4-(4-ethoxy-3-methylphenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-4-oxobutanamide