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2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidine-5-carboxamide
1-(2-methoxy-4-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]isoquinoline-1-carboxamide
(4aS,7aR)-4-(2-methylpropanoyl)-6,6-dioxo-N-phenyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
5-[2-(benzyloxy)ethyl]-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}propanamide
N,N-dimethyl-3-{2-[2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]phenyl}propanamide
2-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1,3-thiazole
3-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(3aR,6aR)-2-(cyclobutylmethyl)-5-[2-(thiophen-2-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-chloro-2-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}quinoline
3-(4-chloro-2-methylbenzoyl)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
1,3-dimethyl-N-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)propyl]-1H-pyrazole-5-carboxamide
4-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1λ6-thiomorpholine-1,1-dione
2-(2,4-dioxoimidazolidin-1-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
N-(1-benzylpiperidin-4-yl)-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-{[6-(3-chloro-4-methoxyphenyl)pyridazin-3-yl]amino}ethan-1-ol
1-(2-chloro-6-fluoro-3-methylbenzoyl)-2-(4-methylpiperazine-1-carbonyl)piperazine
N-[3-(4-methylbenzenesulfonamido)propyl]imidazo[1,2-a]pyridine-6-carboxamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
4-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-1-(3-chlorophenyl)-1H-pyrazole
3-[(2-fluorophenyl)formamido]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
2-(2-methoxyethyl)-9-[2-(3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
8-[(2,5-dimethylphenyl)methyl]-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
N-[2-(2-methoxyphenyl)ethyl]-4-(piperidin-3-yl)benzamide
8-cyclohexyl-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
N-(2-{1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}ethyl)acetamide
4-(1H-1,2,3,4-tetrazol-1-ylmethyl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}benzamide
N-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-oxoethyl)-2-methylpropanamide
4-[5-(1-methoxyethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-3-yl]pyridine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
ethyl 4-(2-chloro-4-{[2-(dimethylamino)ethyl]carbamoyl}phenoxy)piperidine-1-carboxylate
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
3-[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-[3-(4-{methyl[2-(4-methylphenoxy)ethyl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
3-phenyl-N-(1-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
[1-(1-ethyl-1H-indole-5-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
(1S,5R)-3-[(3-chloro-4-methoxyphenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
7-{2-[(1,3-benzothiazol-2-yl)amino]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-ethyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(2-methylprop-2-en-1-yl)butanamide
(3R,4S)-1-(3,4-dimethoxybenzenesulfonyl)-4-(propan-2-yl)pyrrolidin-3-amine
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(1H-1,3-benzodiazol-1-yl)propan-1-one
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-3-propanamidobenzamide
7-cyclopentyl-2-[3-(pyridin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
N-(2-methoxyethyl)-6-(2-methylphenyl)-N-(propan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-methyl-8-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-butyl-N-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide