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5-{4-[4-methyl-2,5-dioxo-1-(thiophen-3-ylmethyl)imidazolidin-4-yl]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl][1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amine
9-methoxy-N-[(2-methoxyphenyl)methyl]-3-[(4-methylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
[(3-chloropyridin-4-yl)methyl](methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
2-[(4aR,7aS)-4-(3-cyclopentylpropanoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
4-{4-[1-butyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]benzoyl}morpholine
5-(3-methoxypropyl)-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-methyl-6-[4-({[1-(phenoxymethyl)cyclopropyl]methyl}amino)piperidin-1-yl]pyrimidin-2-amine
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}ethan-1-one
methyl 1-benzyl-5-{[(4-chlorophenyl)methyl]amino}-3-cyclopropaneamido-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
5-methyl-2-{4-[(4-methyl-3-oxopiperazin-1-yl)methyl]phenyl}-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
7-[cyclohexyl(methoxy)methyl]-4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-cyclopropanecarbonyl-7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(4-tert-butylphenyl)-4-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]butan-1-one
N-methyl-5-oxo-N-(1H-pyrazol-3-ylmethyl)-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
6-(4-fluorophenyl)-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(4-hydroxyphenyl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
2-[(cyclopropylmethyl)sulfanyl]-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]propan-1-one
3-({3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(prop-2-en-1-yl)benzamide
5-fluoro-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1,3-dimethyl-1H-indole-2-carboxamide
6-methyl-5-(5-{[4-(propan-2-yl)phenyl]methyl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(2-methylpiperidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
1-methanesulfonyl-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyridin-4-yl)ethyl]acetamide
11-[(1,3-benzothiazol-2-ylmethyl)amino]-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(1S,5R)-6-(5-fluoro-2-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
8-(6-methylpyridazin-3-yl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-1,3-benzodiazole-4-carboxamide
2-[({5-[1-(2,6-dimethylpyridin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
2-{[2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]amino}-6-methyl-3,4-dihydropyrimidin-4-one
2-(furan-3-carbonyl)-N-(2-methoxyethyl)-1,2,3,4-tetrahydroisoquinoline-8-sulfonamide
naphthalen-1-yl (7R,9aR)-7-[(benzylsulfanyl)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
8-[(5-chloro-2-fluorophenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1-ethyl-1H-pyrazole
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methylpiperazin-2-one
1-(2-fluoro-6-methoxybenzoyl)-3-(3-methoxyphenoxymethyl)piperidine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-(cyclohexylmethyl)piperidine
8-methoxy-2-oxo-N-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-benzyl-8-[(4-methyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecane
3-ethyl-5-{[5-(5-fluoro-2-methylphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazole
ethyl 4-[1-(cyclopent-1-ene-1-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
3-[(2,4-difluorophenyl)methyl]-9-methoxy-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(2S)-2-hydroxy-4-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]butanoic acid