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methyl (2S,4R)-1-methyl-4-(2-methyl-4-phenyl-1,3-thiazole-5-amido)pyrrolidine-2-carboxylate
N-[3-(4-{[2-(1H-1,3-benzodiazol-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-methylfuran-3-carboxamide
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2,2-dimethyl-1-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
1-(2,2-dimethyloxane-4-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 4-{[(2-{1-[1-(furan-2-yl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
methyl 5-(cyclohexylamino)-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)methyl]acetamide
N,N-dimethyl-5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}pyridine-3-carboxamide
1-[3-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidine-1-carbonyl)phenyl]pyrrolidin-2-one
N-cyclopropyl-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
6-methyl-2-{[2-(4H-1,2,4-triazol-4-yl)ethyl]amino}-3,4-dihydropyrimidin-4-one
N-[(2R,3R)-2-methoxy-1'-[(2,3,6-trifluorophenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-4-(4-methylpiperazin-1-yl)benzamide
N-(3-hydroxypropyl)-1-{1-[(2-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-{5-[(2S)-1-(1-benzothiophene-5-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
(1S,5R)-6-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-3-(furan-2-yl)-N-methylbenzamide
4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)piperazin-2-one
6-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carbonitrile
(4aS,7aR)-1-(4-chlorobenzoyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[(4-hydroxy-6-methylquinolin-2-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-cyclopentyl-1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)ethan-1-one
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
1-(5-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
2-(2H-1,3-benzodioxol-5-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}ethan-1-one
N-cyclopropyl-3-{1-[1-(2-fluorophenyl)propan-2-yl]piperidin-4-yl}propanamide
methyl 5-[(8-hydroxyquinolin-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}ethan-1-one
2-ethyl-N-[2-(4-hydroxyphenyl)ethyl]-6-methyl-4-oxo-1-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
1-(furan-2-carbonyl)-4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
1-[cyclohexyl(methyl)amino]-3-[2-(1,4-oxazepan-4-ylmethyl)phenoxy]propan-2-ol
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzonitrile
2-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-(pyrimidin-2-yl)phenol
N-{[7-chloro-2-(2,5-dimethoxyphenyl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]thiophene-2-carboxamide
3-methoxy-1-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]-1,2-dihydropyridin-2-one
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(1-methyl-1H-pyrazole-5-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N,3-diethyl-5-methyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-1,2-oxazole-4-carboxamide
1-(4,6-dimethylquinazolin-2-yl)-N-(3-hydroxy-2,2-dimethylpropyl)piperidine-4-carboxamide
methyl 4-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}benzoate
4-[(1E)-3-[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]prop-1-en-1-yl]-2-methoxyphenol
(1R,9S)-5-amino-12-methyl-3-[2-(thiophen-2-yl)pyrimidin-5-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
2-(dimethyl-1,2-oxazol-4-yl)-N-(1-phenyl-1H-pyrazol-5-yl)pyrrolidine-1-carboxamide
2-[(dimethylamino)methyl]-N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-1,3-thiazole-4-carboxamide
N-(furan-2-ylmethyl)-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidine-4-carboxamide