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1-ethyl-N-[1-(2-methylphenyl)cyclopropyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-{7,9-dioxo-8-azaspiro[4.5]decan-8-yl}-N-[2-(2-methoxyphenyl)ethyl]acetamide
1-{3-[3-(2-methylphenyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
1-(2-phenylethyl)-4-[4-(pyridin-2-yl)pyrimidin-2-yl]piperazin-2-one
1-(2-methylpropyl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}piperidin-4-amine
[(4-fluoro-3-methoxyphenyl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
methyl 2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-6-[(4-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[1-({[(4-phenyl-1,3-thiazol-5-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2H-1,3-benzodioxole-5-carboxamide
7-fluoro-3-{[2-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-(2-chloropyridine-4-carbonyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-({2-[5-(piperidin-1-ylmethyl)thiophen-2-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-[(4-chlorophenyl)methyl]-N-{[(3R,4R)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}benzamide
2-benzyl-N-(6-methylpyridin-3-yl)-1,3-thiazole-4-carboxamide
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl}){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
1-cycloheptyl-N-[(2-methoxynaphthalen-1-yl)methyl]-6-oxopiperidine-3-carboxamide
2-[2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
[1-(2,1,3-benzoxadiazol-5-ylmethyl)-3-benzylpiperidin-3-yl]methanol
1-[(3-fluorophenyl)methyl]-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazine
5-[3-(2-ethylpiperidin-1-yl)-3-oxopropyl]-5-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-one
N-(1-methyl-6-oxopiperidin-3-yl)-2,3-dihydro-1-benzofuran-5-carboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-[(3-methoxyphenyl)methyl]-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
1-(3-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}phenyl)pyrrolidin-2-one
6-(4-methoxyphenyl)-9-[4-(2-oxopyrrolidin-1-yl)benzoyl]-6,9-diazaspiro[4.5]decan-7-one
N-[2-(1H-indol-1-yl)ethyl]-N,3-dimethylfuran-2-carboxamide
1-(carbamoylmethyl)-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
4-(2H-1,3-benzodioxole-5-carbonyl)-1-methylpiperazin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(1-phenylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
N-[5-(2-methyl-4-phenylpiperazine-1-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-7-yl]acetamide
2-(4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)pyrimidine
(1R,5R)-3-cyclobutanecarbonyl-6-(thiophen-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-(4-chlorophenoxy)phenyl]-3-methyl-3-(oxan-4-yl)urea
4-[2-(diethylamino)-2-(furan-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-({methyl[1-(pyridin-4-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
6-ethoxy-2-[1-(2-methoxyethyl)-1H-imidazol-2-yl]quinoline
1-[2-(4-methoxyphenyl)ethyl]-4-[(pyridin-3-ylmethyl)amino]pyrrolidin-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
5-{[(2-amino-5,6-dimethylpyrimidin-4-yl)amino]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
5-[(dimethylamino)methyl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}furan-2-carboxamide
5,7-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(pyridin-3-yl)propan-2-yl]quinoline-4-carboxamide
1-{4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(1H-indazol-1-yl)ethan-1-one
1-(cyclohexylmethyl)-N,N-dimethyl-5-[methyl(1,2-oxazol-3-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl (2S,4S)-4-{[(3-chloro-4-methoxyphenyl)carbamoyl]amino}-1-methylpyrrolidine-2-carboxylate
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-5-ylmethyl)amine