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methyl 3-(butanamidomethyl)-5-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)benzoate
N-{3-[(benzylamino)methyl]-5-(pyrrolidine-1-carbonyl)phenyl}acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(5-propylthiophene-3-carbonyl)piperidine
3-{5-[(2S)-2-acetamido-4-methylpentanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
(2S,3R)-2-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-3-hydroxybutanamide
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-{3-oxo-3-[4-(thiophen-2-ylmethyl)piperazin-1-yl]propyl}pyrrolidin-2-one
(1R,5R)-6-(2-chloro-4,5-difluorobenzoyl)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
2-(3-fluorophenyl)-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}acetamide
1-methyl-4-{3-methyl-5-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}-1,2-dihydroquinolin-2-one
(2S,4S)-4-amino-N-ethyl-1-[2-(2-methoxyphenoxy)acetyl]pyrrolidine-2-carboxamide
N-cyclopentyl-3-{[1-(6-methylpyridin-3-yl)ethyl]sulfamoyl}benzamide
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)furan-2-carboxamide
3-(4-hydroxyphenyl)-N-(5-oxo-1-propylpyrrolidin-3-yl)-1H-pyrazole-5-carboxamide
N-butyl-2-[4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)morpholin-3-yl]acetamide
4-[(2,6-difluoro-3-methylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
2-({[2-(propan-2-yl)pyrimidin-4-yl]methyl}(pyridin-3-ylmethyl)amino)butan-1-ol
2-({2-amino-6-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
1-(1-cyclohexyl-1H-pyrazol-5-yl)-3-[2-(dimethylsulfamoyl)ethyl]urea
2-methoxy-N-[(7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
(1S,5R)-6-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(morpholin-4-yl)-3-[3-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
N-methyl-1-[2-(piperidin-2-yl)ethyl]-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-(2-aminoethyl)-4-[(1R)-1-(4-methoxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-(furan-2-yl)pyrimidine
ethyl 1-(4-methoxy-4-oxobutanoyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrazine-2-carboxamide
2-methoxy-3-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}quinoline
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-propyl-1,3-thiazole-4-carboxamide
2-(dimethylamino)-8-(5-propyl-1,3,4-oxadiazol-2-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-3-phenylpropan-1-ol
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-(4-phenoxybenzoyl)piperidine
1-[(3S,4S)-3-hydroxy-4-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}pyrrolidin-1-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-{[7-(1H-indole-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
2-({[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)amino}methyl)pyridine-3-carboxylic acid
3-methyl-1-[2-(oxolan-3-yl)ethyl]-1,2-dihydroquinoxalin-2-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-ethoxybenzoyl)pyrrolidin-3-yl]methanol
(1-{3-[(pyrimidin-4-yl)amino]propyl}piperidin-2-yl)methanol
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[(4-chlorophenyl)methyl]-5-(3-propyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
2-(difluoromethoxy)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethyl)piperazine
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-3-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
5-[3-(2-methyl-1H-imidazol-1-yl)propyl]-5,6-dihydrophenanthridin-6-one
N-methyl-1-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
(2S,4R)-1-[(4-cyanophenyl)methyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
1-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-4-(4-fluorophenyl)butane-1,4-dione