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(2S,4S)-4-amino-N,N-diethyl-1-[(3-methylphenyl)methanesulfonyl]pyrrolidine-2-carboxamide
3-[(3-hydroxyphenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4,4-difluoropiperidine
8-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(2-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-2-oxoethyl)-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylbenzamide
(2H-1,3-benzodioxol-5-ylmethyl)({[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
2,5-dimethyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
ethyl 4-[(4-chlorophenyl)methyl]-1-[2-(diethylamino)acetyl]piperidine-4-carboxylate
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(3-methylbut-2-enoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-(5-propyl-1,2-oxazole-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-(4-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-one
N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclopropanecarboxamide
2,3-dimethyl-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-1H-indole-7-carboxamide
(1R,7S)-3-[(3-methylphenyl)methyl]-6-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
methyl[(1-{[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
N-ethyl-2-methyl-4-oxo-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[2-(morpholin-4-ylmethyl)propanoyl]piperazin-2-one
3-(1-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1H-imidazol-2-yl)phenol
3,5-dichloro-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}pyridine
5-(3-chloropyridin-2-yl)-8-methoxyquinoline
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
5-tert-butyl-3-{5-[(3,4-difluorophenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrazole
N3-tert-butyl-1-(3-methylbutyl)-4-oxo-N5-[2-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(dimethylsulfamoyl)ethyl]-3-acetamidobenzamide
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-5,6-dimethylpyrimidin-4-amine
ethyl 4-[10-(methoxycarbonyl)-7-oxo-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-3-yl]piperidine-1-carboxylate
N-(2-methoxyethyl)-N-methyl-2-[4-methyl-6-(pyrrolidine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetamide
N-({7-[2-(2-chlorophenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl][(4-methoxyphenyl)methyl](pyridin-2-ylmethyl)amine
methyl 3-(2,3-dimethylbenzoyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2,6-difluoro-3-methylphenyl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
6-ethoxy-4-methyl-2-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1,4-diazepan-1-yl]quinazoline
ethyl 4-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-amido)piperidine-1-carboxylate
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(pyridin-3-yl)ethan-1-one
1-[2-methoxy-4-({[5-(morpholin-4-yl)pentyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-[(2-chloro-5-methylphenyl)formamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]propanamide
5-(1-methylpyrrolidin-3-yl)-3-(1-phenylcyclobutyl)-1,2,4-oxadiazole
4-[(2,4-dimethoxyphenyl)methyl]-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[1-(morpholin-4-ylmethyl)cyclohexyl]-1H-imidazole-2-carboxamide
N-{4-[4-(2-methoxyethoxy)piperidine-1-carbonyl]phenyl}ethane-1-sulfonamide
2-cyclopentyl-9-(2-hydroxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
methyl 1-methyl-2-[3-(1H-pyrazol-3-yl)phenyl]-1H-1,3-benzodiazole-5-carboxylate
2-[(5-methylpyrazin-2-yl)methyl]-9-(morpholine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-1-(6-fluoro-4-methylquinazolin-2-yl)-N-methylpyrrolidine-2-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(pyrazin-2-yl)propanamide
N-methyl-3-[(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)methyl]-1,2,4-oxadiazole-5-carboxamide