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3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
methyl 4-{[3-(1-acetamido-3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}benzoate
3,4-dimethoxy-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
(1-benzothiophen-2-ylmethyl)(methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[2-(dimethylamino)ethyl]-N-ethyl-1,2-oxazole-3-carboxamide
2-[2-(3-ethyl-2-imino-2,3-dihydro-1H-1,3-benzodiazol-1-yl)acetamido]-N,N-dimethylpropanamide
1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
methyl 2-({1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)acetate
8-(3-acetyl-1H-pyrazole-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[4-({3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenoxy]pyrimidine
1-{2-fluoro-3-[4-(4-methylpiperazin-1-yl)quinazolin-6-yl]phenyl}ethan-1-one
7-(1H-1,3-benzodiazole-5-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(1-cyclobutylpiperidin-4-yl)oxy]-N-cyclopropyl-4-methoxybenzamide
3-(5-methylfuran-2-yl)-N-[(4-phenylmorpholin-2-yl)methyl]-1H-pyrazole-5-carboxamide
(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
4-{[(2-hydroxyethyl)(thiophen-2-ylmethyl)amino]methyl}benzonitrile
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
2-chloro-4-fluoro-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[3-(pyridin-3-yloxy)propyl]-1H-1,3-benzodiazole-7-carboxamide
2-[2-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-5,6-dimethyl-2,3-dihydropyridazin-3-one
1-(3-fluoro-2-methoxybenzoyl)-3-(3-methoxybenzoyl)piperidine
(1S,3R)-3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]cyclohexan-1-amine
N-[(3S,4R)-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
1-[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(2H-indazol-2-yl)ethan-1-one
2-({1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
(2R,3R,6R)-5-(6-ethylpyrimidin-4-yl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
8-(2,2-dimethylpropyl)-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(7-butanoyl-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-3-carboxamide
1-(2-methylpyridin-4-yl)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,4-diazepane
3-(cyclopropylmethyl)-5-{imidazo[1,2-a]pyrimidin-2-yl}-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
(1r,4r)-4-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine-1-carbonyl}cyclohexan-1-ol
1-(4-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
(2S,4R)-4-amino-1-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-(3-methoxyphenoxy)-N-[2-(4-methylphenyl)propan-2-yl]acetamide
ethyl (2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(4-methyl-1H-pyrazol-1-yl)propanamide
3-[3-(1H-imidazol-2-yl)propyl]-1-(6-methoxypyridin-3-yl)urea
1-{1'-[(1-ethyl-1H-imidazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
(3R,7S,8aS)-7-(benzylamino)-3-[(1S)-1-hydroxyethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
methyl 3-(2H-1,3-benzodioxol-4-ylmethyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[methyl(piperidin-4-yl)sulfamoyl]-N-(1,2-oxazol-3-ylmethyl)benzamide
4-(benzyloxy)-1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
ethyl 4-{[6-chloro-4-(4-methoxypiperidin-1-yl)quinazolin-2-yl]methyl}piperazine-1-carboxylate
4-[4-(methylamino)benzoyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(pyridin-3-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]-2-(pyrrolidin-1-yl)acetamide
6-(morpholin-4-yl)-N4-[2-(phenylamino)ethyl]pyrimidine-2,4-diamine
(1R,5R)-6-[(5-methylfuran-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-4-yl)-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione