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N,N-dimethyl-2-[(1S,5R)-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
1-(2-methoxyethyl)-4-[6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperazine
N-[(2-methylphenyl)methyl]-4-(4-methylpiperazin-1-yl)-N-(prop-2-en-1-yl)pentanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-methyl-4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]acetamide
4-{4-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]piperidin-1-yl}-N-cyclopentylbenzamide
N-methyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
3-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}-1-(pyrrolidin-1-yl)propan-1-one
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[2-(3,4-dimethoxyphenyl)ethyl]-1-methylurea
4-fluorophenyl (7R,9aR)-7-benzyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
6-methyl-3-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1,4-dihydroquinolin-4-one
3-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1,2-benzoxazole
(1S,5R)-3-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(1-propyl-1H-1,2,3-triazol-4-yl)urea
5-methyl-2-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}furan-3-carboxamide
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-phenylpiperazin-2-one
2-(2-{[ethyl(oxan-4-yl)amino]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
N-[(3,4-dimethoxyphenyl)methyl]-2-(4-methylpiperazin-1-yl)-6-(thiophen-3-yl)pyridine-3-carboxamide
4-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-6-ethyl-1,2-dihydropyridin-2-one
2-(cyclopent-2-en-1-yl)-1-{4-[(1,2-oxazol-3-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
5-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,4-dimethylpyrimidine
3-[({[3-(cyclopentyloxy)phenyl]carbamoyl}amino)methyl]-N,N-dimethylbenzamide
(2S,3R)-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methyl-2-(methylamino)pentan-1-one
(2S,4R)-N-cyclopropyl-1-[(4-ethylphenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
3-[4-(benzyloxy)piperidin-1-yl]-5-(3-methoxyphenyl)-1,2,4-triazine
3-(3-chloro-1,2-oxazol-5-yl)-1-[2-(furan-2-yl)azepan-1-yl]propan-1-one
2-(3-chloro-5-fluorophenyl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]ethan-1-one
3-{[(6-chloroquinolin-2-yl)methyl](methyl)amino}propane-1,2-diol
3-[(2R,3R,6R)-5-(6-methoxypyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
methyl 4-[(2-{[2-(1,3-thiazol-2-yl)piperidin-1-yl]methyl}quinazolin-4-yl)amino]butanoate
1-(2,6-dimethylpyridin-4-yl)-4-(1-propylpiperidin-4-yl)piperazine
5-amino-3-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-(2-methyl-1H-pyrrole-3-carbonyl)-4-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-1,4-diazepan-6-ol
7-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
1-(3-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-8-methylimidazo[1,2-a]pyridine-2-carbonyl)piperidine
2-ethyl-9-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenyl-2,9-diazaspiro[5.5]undecane
6-(2,6-dimethylquinoline-4-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[(6-methylpyridin-2-yl)methyl]acetamide
(3S,4S)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]benzene-1,3-diol
2-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-5-(2-methylpropyl)-1,2,4-oxadiazole
2-{9-[(4-ethoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
(2S,4R)-1-[(2,5-dimethylphenyl)methyl]-N,N-dimethyl-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carboxamide
N-[3-(4-chlorophenoxy)-2-hydroxypropyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(2-phenoxyethyl)piperazine
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-1-methyl-3-propyl-1H-pyrazole
N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-methylpiperazin-2-one
4-methoxy-N-(2-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
(2R,3R)-1'-methanesulfonyl-3-(thiomorpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol