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6-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]pyridine-2-carbonitrile
3-(2-methylpropyl)-5-[1-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
(1S,5R)-N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-10-oxo-3,9-diazabicyclo[3.3.2]decane-3-carboxamide
2-(3-benzoylpiperidin-1-yl)-4-(pyrrolidine-1-carbonyl)pyridine
2-methoxy-N-{2-methyl-1-[7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}acetamide
3-[(2-methoxyethyl)sulfamoyl]-5-(quinolin-8-yl)benzoic acid
2-(3-fluorophenyl)-N-({7-[(8-methoxyquinolin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
1-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-(pyridin-4-yl)propan-1-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(methylsulfanyl)acetamide
1-cyclopentyl-4-[4-(pyridin-4-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
2-[(2-chlorophenyl)methyl]-4-(thiophene-3-sulfonyl)morpholine
3-butanamido-N-ethyl-N-(pyridin-2-ylmethyl)benzamide
4-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,4-oxazepane
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
{3-[(3-chlorophenyl)methyl]-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methanol
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-ethyl-2-methylpyrimidin-4-amine
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[3-(pyridin-3-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-4-(3-methylphenoxy)piperidine
(3S,4S)-1-(4-methoxybenzoyl)-4-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrrolidin-3-ol
3-(2-methoxyphenyl)-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)propanamide
5-chloro-4-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-2-methoxyphenol
1-cyclopentyl-3-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]piperidine
4,6-dimethyl-1-{2-[4-(piperidin-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
2,6,8-trimethyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}quinoline-4-carboxamide
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
9-(1-phenyl-1H-pyrazol-5-yl)-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
2-(2-methylpropyl)-6-(2,4,5-trimethoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-methoxy-N-{1-[1-(2-methoxyacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
(3S,4S)-4-(4-fluorophenyl)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidin-3-ol
(4aS,8aR)-2-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-decahydroisoquinoline
N-({4-[(4-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-3-ylmethyl)-1,2,5-thiadiazole-3-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-{3-methyl-3H-imidazo[4,5-b]pyridin-2-yl}propanamide
methyl 3-(2H-1,3-benzodioxol-4-ylmethyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)pyridine
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(1-ethyl-1H-imidazol-2-yl)-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
2-(8-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl)acetic acid
5-fluoro-2-[1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(1H-pyrazol-1-yl)benzamide
4-acetyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-1,4-diazepane-1-carboxamide
2-amino-4-[3-(difluoromethoxy)phenyl]-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
2-[2-(dimethylamino)ethyl]-8-[2-(pyridin-2-ylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(2-methylpropyl)cyclopropyl]-4-(1H-pyrazol-4-yl)butanamide
3-({3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}methyl)-1-methyl-1,2-dihydroquinolin-2-one
1-[2-(dimethylamino)ethyl]-4-[3-(4-fluorophenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
1-(4-methoxyquinoline-2-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[1-({[(2-methyl-1,3-thiazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
methyl 2-[1-benzyl-8-(butan-2-yl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
2-[(3-fluorophenyl)methyl]-4-{4-[(3-hydroxy-4-methoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione