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4-methyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
2-[1-(1-cyclopropylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-methyl-1H-imidazole
1-[(4-methoxyphenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-{[(3R,4R)-4-hydroxypyrrolidin-3-yl]amino}-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
3-(4-phenoxybenzoyl)-1-(thiophene-2-carbonyl)piperidine
(4aR,7aS)-1-(2-methoxyacetyl)-4-(quinoxaline-6-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]-N-methylpyrimidin-2-amine
3-[(tert-butylamino)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
5-(3-ethyl-5-methyl-1,2-oxazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[(2-chlorophenyl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-4-yl]-1-[2-(piperidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
N-[(3-fluorophenyl)methyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[3-(morpholin-4-yl)propyl]acetamide
2-[1-(6-methoxypyridin-2-yl)-4-methyl-1H-1,3-benzodiazol-2-yl]ethan-1-ol
N,N-dimethyl-2-{[4-(1H-1,2,4-triazol-1-yl)butanamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-methoxy-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine
[2-methyl-2-(morpholin-4-ylmethyl)propyl](pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
3-(4-{1-[(4-ethylphenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)propanamide
3-(1H-imidazol-1-ylmethyl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperidine
N-[2-(1,3-benzothiazol-2-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
(2S,4S)-4-{4-[2-(3-methylbut-2-enamido)propan-2-yl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxylic acid
N-[(2R,3R)-1'-{[4-(difluoromethoxy)phenyl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-6-[(thiolan-3-yl)amino]pyridine-3-carboxamide
5-(furan-2-ylmethyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine
5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1-(2-methoxyethyl)piperidin-2-one
4-[(5-chloro-2-hydroxyphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-N-(3,5-dimethylphenyl)-3-oxopropanamide
9-(5-acetylpyridin-2-yl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-(but-2-yn-1-yl)-5-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
N-(2-{4-[(4-phenylpiperazin-1-yl)methyl]phenoxy}propyl)-2-(piperidin-1-yl)acetamide
2-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-4-carbonitrile
6-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)imidazo[1,2-a]pyridine-2-carboxamide
2,3-dimethyl-5-{3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}benzene-1-sulfonamide
1-(2H-1,3-benzodioxole-5-carbonyl)-4-{2-[(2-methylphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[(3-methylpyridin-4-yl)methyl]amino}methyl)piperidin-2-one
(1S,5R)-6-[(5-chlorothiophen-2-yl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(6-methyl-2-propylpyrimidin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
3-[2-(3-acetylpiperidin-1-yl)-2-oxoethyl]-1-benzyl-3-(2-methylphenyl)pyrrolidine-2,5-dione
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(2-methyl-1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-2-(oxan-4-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
1-{1-[5-(hydroxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-phenylethan-1-ol
3-methyl-N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide