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3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-5-(2-methylpropyl)-1H-pyrazole
1'-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-{[4-(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]oxy}acetic acid
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
ethyl 1-({3-[2-hydroxy-3-(morpholin-4-yl)propoxy]phenyl}methyl)piperidine-4-carboxylate
N-{[2-(3-chlorophenyl)-7-fluoroquinolin-3-yl]methyl}-4-methoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
1-(2-{[(3,5-difluorophenyl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
1-(3-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylsulfanyl)ethan-1-one
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pentanamide
2-amino-8-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[3-(1H-imidazol-1-yl)propyl]-2-(2-methoxy-3,5-dimethylphenyl)-1H-imidazole
cyclopentyl 4-({[(5-methylpyrazin-2-yl)methyl]carbamoyl}amino)benzoate
N-[(2R,3R)-2-methoxy-1'-[2-(3-methoxyphenyl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
4-(hydroxymethyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}azepan-4-ol
4-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
({3-[2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-2-yl)ethoxy]phenyl}methyl)(methyl)(quinolin-8-ylmethyl)amine
8-(2,2-diethylcyclopropanecarbonyl)-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
methyl 3-(4-methyl-2-oxopentanoyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[5-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
ethyl 5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
4-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidin-2-amine
3,5-difluoro-N-{[8-(2-phenylacetyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
8-(cyclopropylmethyl)-N-[(4-methylphenyl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
6-[1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
1-(4-{[(dicyclopropylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
3-ethyl-1-{[1-(1H-indol-2-ylmethyl)piperidin-4-yl]methyl}urea
1-(3-chloro-2-propoxyphenyl)-3-[2-(ethanesulfonyl)ethyl]urea
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-methyl-3-(5-phenyl-1,3,4-thiadiazol-2-yl)urea
5-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-(5-chloro-2-methoxyphenyl)-3-[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-3-yl]propanamide
3-[(2,3-dimethoxyphenyl)methyl]-5-methyl-5-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-methylfuran-3-carboxamide
5-{[3-cyclopropyl-1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}-2-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
1-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-3-(4-methoxy-3,5-dimethylphenyl)urea
2-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-5-methylpyrimidin-4-amine
7-fluoro-2-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
N4-{imidazo[1,2-a]pyridin-2-ylmethyl}-6-methoxypyrimidine-2,4-diamine
1-(5-{[butyl(methyl)amino]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]pyrrolidin-2-one
ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
2-methoxy-N-[(2R,3R)-1'-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-{[4-(methoxymethyl)piperidin-1-yl]methyl}-5,8-dimethylquinolin-4-ol
1-{[1-(2-amino-5-ethylpyrimidin-4-yl)piperidin-4-yl]methyl}pyrrolidin-2-one
(3-ethyl-1-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)methanol
4-oxo-N-(5-oxo-1-propylpyrrolidin-3-yl)-3,4-dihydroquinazoline-2-carboxamide
7-fluoro-2-methyl-4-{4-[2-(pyrrolidin-1-yl)ethyl]piperazine-1-carbonyl}quinoline