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(2S,4R)-4-{[(2,5-dimethylphenyl)methyl]amino}-N,1-bis(propan-2-yl)pyrrolidine-2-carboxamide
4-(cyclopentylsulfamoyl)-N-(1H-imidazol-2-ylmethyl)benzamide
2-{[3-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}benzonitrile
1-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]cyclopropan-1-amine
3-(2-benzyl-3-oxopiperazin-1-yl)-N-(2,4-dimethylphenyl)-3-oxopropanamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl][(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[3-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]methanol
4-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidin-3-yl]-2-(pyridin-4-yl)pyridine
3-(1-methyl-1H-pyrazol-5-yl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]propanamide
5-[4-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)phenoxymethyl]furan-2-carboxylic acid
1-[(3,5-dimethylphenyl)methyl]-4-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperazin-2-one
6-cyclopropyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrimidin-4-amine
N-[(3-chlorophenyl)methyl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
4-[(5-{1-[(3-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
1-{2-[1-(2-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[3-(morpholin-4-yl)propyl]amine
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[4-(1H-pyrazol-1-yl)butan-2-yl]propanamide
6-methyl-1-[2-(methylsulfanyl)phenyl]-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-one
7-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-1H-1,3-benzodiazole
5-(3-methylbutyl)-5-{1-[4-(propan-2-yloxy)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
3-[3-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
4-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)pyridine
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]pyridine-2-carboxamide
8-methyl-N-(4-methyl-2-oxo-1,2-dihydroquinolin-7-yl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
3-ethyl-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidine-3-carboxylic acid
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[2-(3-fluorophenyl)ethyl]piperidine-4-carboxamide
2-methyl-6-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
1-[(4-butoxyphenyl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-{[4-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-methoxy-N-methylbenzamide
N-cyclopentyl-4-(4-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}piperidin-1-yl)benzamide
(3S,4R)-4-(2-methoxyphenyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidine-3-carboxylic acid
3-[(3-fluorophenyl)methyl]-N-methyl-N-(thiophen-2-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
3-(diphenylmethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
(3aR,7aS)-5-methyl-2-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
5-{[(methylcarbamoyl)methyl]carbamoyl}-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxylic acid
N-cyclopropyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-[(prop-2-en-1-yl)amino]benzamide
N-tert-butyl-3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
7-[4-(2-methyl-1H-imidazol-1-yl)butanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
3-(dimethylamino)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-2-(4-methoxypiperidin-1-yl)pyridine
2-(5-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-3-yl}-1-(2-methylphenyl)-1H-1,2,4-triazol-3-yl)acetamide
1-(2,3-dihydro-1-benzothiophene-2-carbonyl)-4-methanesulfonyl-1,4-diazepane
2-[3-(2,6-dimethoxyphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(3-methylphenoxy)piperidine
2-[(4-methoxyphenyl)amino]-2-methyl-N-[(1-methylpiperidin-3-yl)methyl]propanamide
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine