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N-[(5-chlorothiophen-2-yl)methyl]-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
5-(2-chlorophenyl)-4-[1-(2,5-dimethylbenzoyl)piperidin-3-yl]pyrimidine
1-[2-(dimethylamino)ethyl]-3-(1-methyl-1H-indazol-6-yl)-1-(oxolan-2-ylmethyl)urea
2,2-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrrolidin-3-amine
ethyl 4-[(4-methoxyphenyl)methyl]-1-(3-methoxypropanoyl)piperidine-4-carboxylate
4-chloro-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1H-pyrazole-3-carboxamide
N-(3-chloro-4-fluorophenyl)-3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}propanamide
2-{3-oxo-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-2-yl}-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
3-[3-(methylsulfanyl)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(1-methylpiperidin-3-yl)ethyl]-3-(1,2-oxazinan-2-yl)propanamide
({3-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)(methyl)(1,2-oxazol-3-ylmethyl)amine
{4-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]morpholin-3-yl}methanol
2-phenoxy-N-[2-(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
3-(1-cyclopropanecarbonylpiperidin-4-yl)-3,9-diazaspiro[5.5]undecane
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
({4-cyclopropyl-5-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
7-chloro-3-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-indole
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-phenylacetamide
(3S,4R)-1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
{1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
1-[(1R,5S,6R)-6-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]butan-1-one
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-(2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1-{[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
8-(furan-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[3-(1H-imidazol-2-yl)piperidin-1-yl]quinoxaline
2,6-dimethyl-4-[({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)methyl]phenyl acetate
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(furan-2-yl)propanamide
6-({[(5-chloro-2-ethoxyphenyl)methyl](methyl)amino}methyl)-1,4-oxazepan-6-ol
N-[(3,4-difluorophenyl)methyl]-5-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
8-(furan-3-ylmethyl)-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
4-methoxy-2-{[methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
N-(6-phenoxypyridin-3-yl)-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-4-carboxamide
3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
N-{[1-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)piperidin-4-yl]methyl}acetamide
N-butyl-1-[1,3-dioxo-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-4-carboxamide
(3-{4-[1-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}phenyl)methanol
N-methyl-N-(2-{2-[2-(5-methylfuran-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)methanesulfonamide
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-propanoyl-1,4-diazepan-2-one
5-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-methyl-1H-pyrazole-4-carboxamide
N-(1-methoxypropan-2-yl)-1-[2-(2,3,6-trimethylphenoxy)acetyl]piperidine-4-carboxamide
N-[2-(adamantan-1-yl)ethyl]-1-ethyl-N-methyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-7-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
(1R,5R)-6-benzyl-3-(1,3-thiazol-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(5-fluoro-2-methylphenyl)methyl]propanamide