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1-(5-ethyl-1,3,4-thiadiazol-2-yl)-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
ethyl 5-(1-ethyl-1H-pyrazole-4-carbonyl)-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}propanamide
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-3-{[(2-hydroxyethyl)amino]methyl}-1-(2-phenylethyl)piperidin-2-one
2-(3-hydroxypiperidin-1-yl)-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)acetamide
3-[2-(dimethylamino)ethyl]-1-ethyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(4-methylphenyl)-2-(pyrrolidin-1-yl)pyrimidin-5-yl]benzamide
1-cyclobutanecarbonyl-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
8-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
N-(2-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-2-oxoethyl)acetamide
8-[(2,5-difluorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-fluoro-4-methylbenzenesulfonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-2,4-dimethoxy-N-(pyridin-3-ylmethyl)benzamide
N-ethyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-4-ylmethyl)propanamide
8-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(thiophen-3-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
ethyl 2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-2-yl]acetate
(3S,4R)-4-(4-fluorophenyl)-1-{2-[methyl(phenyl)amino]acetyl}pyrrolidine-3-carboxylic acid
2-methyl-5-(3-methylphenyl)-4-{1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-3-yl}pyrimidine
4-[4-(3,5-difluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-methylpiperidin-4-ol
3-(3-hydroxyquinoxalin-2-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}propanamide
1-methyl-6-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-indole
1-[(3,5-difluorophenyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
2,4-difluoro-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-5-chloro-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-[4-(methylsulfanyl)phenyl]acetic acid
1-methyl-4-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]ethyl}piperazine
1'-[(7-hydroxyquinolin-3-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(4S)-3-{2-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-phenyl-1,3-oxazolidin-2-one
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
(1S,5R)-3-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-3,9-diazabicyclo[3.3.2]decan-10-one
2-benzyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-1,3-benzoxazole
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-[2-(1H-indol-3-yl)ethyl]-1-methylpyrrolidine-3-carboxamide
2-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)ethan-1-amine
N-[(1-{[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]acetamide
2-[(1H-1,3-benzodiazol-2-ylmethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]ethan-1-ol
1-[(2-chlorophenyl)methyl]-N-methyl-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-[(2R,3R)-2-hydroxy-1'-[(3-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
4-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
1-(2-chlorophenyl)-2-{[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}ethan-1-ol
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidine
2-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
4-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
6-[(3-fluorophenyl)methyl]-2-[3-(morpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
(2,1,3-benzoxadiazol-5-ylmethyl)(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)amine
(4aS,7aR)-1-(3-hydroxybenzoyl)-4-[(5-methylfuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide