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2-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
3-[2-(hydroxymethyl)phenyl]-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
4-methyl-5-{1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
1-methyl-9-(prop-2-en-1-yl)-4-[2-(4H-1,2,4-triazol-4-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(naphthalen-2-yloxy)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]propanamide
3-(ethoxymethyl)-1-methyl-5-{[(4-methyl-1,3-thiazol-2-yl)sulfanyl]methyl}-1H-1,2,4-triazole
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
ethyl 1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(methylsulfanyl)benzamide
8-[(4-acetylphenyl)methyl]-3-[3-(dimethylamino)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(2-aminopyridin-3-yl)methyl]-4-(pyridin-4-yl)-1,4-diazepan-6-ol
3-(2,5-difluorobenzoyl)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
5-butyl-1'-(5-methyl-1,2-oxazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 1-{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carboxylate
1-cyclopentyl-3-(3-methoxyphenyl)-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
methyl 3-(furan-2-amido)-5-{[(5-methyl-3-phenyl-1,2-oxazol-4-yl)formamido]methyl}benzoate
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-[(4-methylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1-ethyl-1H-pyrazol-4-yl)-4-(3-methylphenyl)-4H-1,2,4-triazole
6-(pyrrolidin-1-ylmethyl)-4-[4-(trifluoromethyl)pyrimidin-2-yl]-1,4-oxazepan-6-ol
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
1-(3,4-dichlorophenyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperazine
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
4-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)-1-(2-methoxyethyl)pyrrolidin-2-one
methyl 3-[2-(2-fluorophenyl)acetamido]-6-{[methyl(propan-2-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
3-(1,4-diazepane-1-sulfonyl)-N-(1,4-dioxan-2-ylmethyl)benzamide
(3aS,6aS)-2-[(4-methylphenyl)methyl]-5-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-ethyl-3-methyl-N-(5-methyl-2-pentanamidophenyl)-1H-pyrazole-5-carboxamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
2-[(3,5-difluorophenyl)methyl]-8-(2-ethoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3,4-dimethoxyphenyl)methyl]-4-methoxy-N-(pyridin-4-ylmethyl)benzamide
(2R,6S)-4-(1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-2,6-dimethylmorpholine
1-(cyclohexylmethyl)-5-{[2-(4-methoxyphenyl)ethyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N,2-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyrimidine-3-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
(2R,3R)-3-amino-1'-(quinoline-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[5-(quinolin-8-yl)-1H-indol-1-yl]acetamide
4-[5-({5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}methyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]-3-methylpyridine
4'-{[2-(difluoromethoxy)phenyl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(3-methoxyphenoxymethyl)-N-(2-methoxyphenyl)piperidine-1-carboxamide
2-[(5-chlorothiophen-2-yl)methyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
(3S,5S)-1-cyclohexyl-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-{[7-(2-chloro-6-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
5-(3-fluorophenoxymethyl)-N-[2-hydroxy-1-(pyridin-3-yl)ethyl]-1H-pyrazole-3-carboxamide
3-methyl-1-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)butan-1-ol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
ethyl(methyl){[(2R,5S)-5-[(1-methyl-1H-indazol-5-yl)methyl]oxolan-2-yl]methyl}amine
2-methyl-3-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)quinoxaline
9-[(2-chloro-5-fluorophenyl)methyl]-2-cyclopentyl-2,9-diazaspiro[5.5]undecan-3-one