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(4aS,8aR)-1-(2-phenylethyl)-6-(pyridin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
3-[5-(2,4-dimethoxybenzoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
2-[(furan-2-ylmethyl)({[4-methoxy-3-(methoxymethyl)phenyl]methyl})amino]butan-1-ol
2-(2-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}ethyl)pyridine
1-ethyl-4-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amino]methyl}-1H-pyrrole-2-carbonitrile
3-{1-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}-4-methoxyphenol
1-[(4aR,8aR)-4a-hydroxy-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-2-yl]-2-(pyridin-3-yl)ethan-1-one
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-(2-methylpropyl)piperidin-4-yl]acetate
4-(5-phenyl-1,3,4-thiadiazol-2-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2,6-dimethoxy-3-[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]pyridine
1-[1-(4-benzylpiperazine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]-2-(2-chloro-4-fluorophenyl)ethan-1-one
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-2,8-diazaspiro[4.5]decane-3-carboxamide
2-({[(3R,4R)-1-[(3,5-difluoro-4-methoxyphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
[4-(4-{1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}pyridin-2-yl)phenyl]methanol
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2,3-dimethylphenyl)carbamoyl]piperidine-4-carboxylate
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
2,4-dimethoxy-6-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrimidine
2-(dimethyl-1,2-oxazol-4-yl)-1-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]ethan-1-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N,5-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-cyclopentyl-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]acetamide
methyl 2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
1-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
4-(2-chlorophenoxy)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N-[2-(diethylamino)ethyl]-N-ethylacetamide
N-(2,4-dimethylphenyl)-3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
N4-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
3-[1-(1-cyclohexylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(3-fluorophenyl)urea
3-(aminomethyl)-4-(2-phenoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-acetamido-1-(oxolan-2-ylmethyl)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(4-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)furan-2-carboxamide
5-(2-methylphenyl)-4-{1-[2-(methylsulfanyl)benzoyl]piperidin-3-yl}-2-(pyridin-4-yl)pyrimidine
[(2-ethylphenyl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4,4,4-trifluorobutan-1-one
5-[3-(3-fluorophenoxy)azetidine-1-carbonyl]-1H-1,2,3-triazole
(1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperidin-4-yl)methanol
3-ethyl-N,4-dimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-pyrazole-5-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propanamide
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
N-(2-methoxyethyl)-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)furan-2-carboxamide
N-cyclohexyl-5-{1-[(dimethylsulfamoyl)amino]ethyl}-N,4-dimethylpyrimidin-2-amine
1-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
3-(2,3-dihydro-1H-isoindol-2-yl)-N-(1-ethyl-4-methyl-1H-pyrazol-5-yl)propanamide
1-benzyl-N3-cyclopropyl-N5-[(3,4-difluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(3,5-dimethylphenyl)-4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
N-cyclopropyl-1-(2-{1-[(6-methylpyridin-2-yl)methyl]piperidin-2-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
2-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]-5-methylpyrazine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(4,6-dimethylpyrimidin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid