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5-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(1-methanesulfonylpiperidin-4-yl)-N-(2-phenylethyl)piperidine-3-carboxamide
1-{3-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-3-ethyl-4-methylpiperidin-4-ol
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]oxolane-3-carboxamide
N-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-(3-methoxyphenyl)-4-[2-(pyrrolidin-3-yl)benzoyl]piperazin-2-one
1-benzyl-6-(cyclopropylmethoxy)-4-(pyrazine-2-carbonyl)-1,4-diazepan-2-one
1-{4-[(2-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-methylbutan-1-ol
(3S,9aR)-8-(3-phenylpropyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-(morpholin-3-yl)ethan-1-one
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-[(1-methylpyrrolidin-3-yl)methyl]benzene-1-sulfonamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-methyl-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]urea
4-methyl-2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-7-(methylsulfanyl)quinoline
2-{4-[(2-chlorophenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(2,3-dihydro-1H-inden-2-yl)-N,1-dimethyl-1H-1,2,3-benzotriazole-5-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(2-propoxyethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
ethyl 3-[(3-chlorophenyl)methyl]-1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxylate
6-(piperidin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
5-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(oxolan-2-ylmethyl)propanamide
methyl 4-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentanoate
N-[(2-phenoxypyridin-3-yl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
N-ethyl-2-(7-methyl-2-oxo-2H-chromen-4-yl)-N-(oxolan-2-ylmethyl)acetamide
4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-methylpiperazin-2-one
1-(6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-2-yl)ethan-1-ol
3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-[1-(furan-2-ylmethyl)piperidin-4-yl]urea
5-(3-methoxyphenyl)-3-{4-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}-1,2,4-triazine
(3R,5S)-1-benzyl-N-[2-(dimethylamino)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
1-cyclopropyl-N-[2-(2,3-dimethoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
2-(5-{[6-(dimethylamino)pyridin-3-yl]methyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
N-methyl-4-[2-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
3-(3,5-dimethylphenyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-4,4,4-trifluorobutan-1-one
2,5-dimethoxy-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
3-{1-[2-(2-fluorophenyl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2,3,5-trimethyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
[(3R,4S)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
9-(2,6-dimethoxybenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)furan-2-carboxamide
1-cyclopentyl-4-(2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazin-2-one
(1S,5R)-N,N-dimethyl-6-[(5-methylthiophen-2-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]acetamide
[1-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
3-ethyl-1-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-1H-pyrazole-5-carboxamide
3-{3-[3-(4-chlorobenzoyl)piperidin-1-yl]-3-oxopropyl}-3,4-dihydroquinazolin-4-one
(3R,4R)-N-[2-(2-fluorophenyl)ethyl]-3-hydroxy-3,4-dimethylpyrrolidine-1-carboxamide
2-[1-(2-methyl-2-phenylpropanoyl)pyrrolidin-3-yl]benzoic acid