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N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]propanamide
8-[(2-cyclohexylpyrimidin-5-yl)methyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-[(1R,2R)-2-acetamido-2,3-dihydro-1H-inden-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)naphthalene-1-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-4-[3-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-methoxy-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-4-({8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-1H-pyrazole
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(ethyl)({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amine
N-methyl-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
N-({7-[4-(dimethylamino)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-N-(2-methoxyethyl)-6-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[4-(1H-indol-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2-phenylethan-1-ol
2-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)-N-methylethane-1-sulfonamide
5-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-yl}-1-methyl-1H-1,2,4-triazole
4-{[2-(morpholin-4-yl)ethyl]amino}pyrimidine-5-carboxylic acid
3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-[(2E)-3-phenylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
[2-({4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
4-fluoro-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methylbenzamide
8-[(2,3-difluoro-6-methoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-9-(3-methyl-1H-pyrazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(5S,9aS,9bS)-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-(8-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]acetyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl)acetic acid
3-{1-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-4-phenyl-1H-imidazol-5-yl}phenol
4-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-methoxybenzamide
1-(3-methoxypropyl)-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
ethyl 4-{[4-(3-chloro-4-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
2-methyl-9-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
7-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-ethyl-3-methyl-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
4-[(1-propyl-1H-imidazol-2-yl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(2-methoxyphenyl)methyl]acetamide
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
6-methoxy-N4-methyl-N4-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine
3-hexyl-8-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{[(thiophen-2-ylmethyl)carbamoyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-{[1-(2-hydroxyethyl)piperidin-3-yl]methyl}-2-(4-methoxyphenyl)acetamide
1-[4-(2-benzylmorpholin-4-yl)-4-oxobutyl]pyrrolidin-2-one
3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-(propan-2-yl)piperidine-1-carboxamide
1-[(3-methylphenyl)methyl]-4-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-phenylpyrrolidin-3-ol
N-(2,3-dihydro-1H-inden-1-yl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
4-(azepan-1-yl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-4-oxobutanamide
2-[4-(4-benzylpiperazine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]-4-(furan-2-yl)pyrimidine
5-methyl-N-{4-[2-(pyridin-4-yl)-1H-imidazol-1-yl]phenyl}furan-3-carboxamide
2-[(3-chlorophenyl)methyl]-N-ethyl-N-(2-hydroxyethyl)-1,3-benzoxazole-6-carboxamide