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1-cyclopropyl-N-methyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-6-oxopiperidine-3-carboxamide
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
8-(3-methoxypropyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyridine-2-carbonitrile
methyl[2-(pyridin-2-yl)ethyl](2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
(3R)-1-(2,6-difluoro-4-methoxybenzoyl)-3,4,4-trimethylpyrrolidin-3-ol
2-(3-{[4-(aminomethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-[(2-methylphenyl)methyl]piperazine
4-propyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-5-carboxamide
N-(1-benzothiophen-2-ylmethyl)-4-methyl-5-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
3-chloro-N-ethyl-N-[2-(pyrrolidin-1-yl)ethyl]thiophene-2-carboxamide
3-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-N-[(2-fluorophenyl)methyl]propanamide
N-[(2R,3R)-2-hydroxy-1'-[(4-hydroxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
1-methyl-N-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}-1H-indole-6-carboxamide
1-benzyl-8-[(2,6-difluorophenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,4S)-2-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-2-azabicyclo[2.2.1]heptane
ethyl 5-({3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}methyl)furan-2-carboxylate
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
N-[2-methyl-4-(2,3,4-trimethoxyphenyl)phenyl]pyridine-3-carboxamide
4-acetamido-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}butanamide
4-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1-phenylpiperazin-2-one
1-(2-chloropyridine-4-carbonyl)-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
2-(5-acetylthiophen-3-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
(2S,3R)-3-hydroxy-2-{[5-(2-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}butanamide
N-(2,2-diphenylethyl)-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-{2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridine-4-carbonyl}morpholine
methyl 3-{[5-(methoxymethyl)furan-2-yl]methyl}-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
(1S,5R)-3-acetyl-N-(3,4-dimethylphenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-(hydroxymethyl)-N-[(3-propoxyphenyl)methyl]-1H-1,3-benzodiazole-5-carboxamide
5-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)thiophene-3-carboxamide
4-[(dimethylsulfamoyl)amino]-1-(2-phenylethyl)pyrrolidin-2-one
3-{[2-(2-phenylethyl)morpholin-4-yl]methyl}-1,2-dihydroquinolin-2-one
N-(2-hydroxyethyl)-N-methyl-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
methyl 3-(1-ethyl-1H-pyrazole-4-carbonyl)-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
N-methyl-N-(1,3-thiazol-2-ylmethyl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
N-[1-(dimethylamino)-2-methylpropan-2-yl]-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
N-(2-hydroxybutyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyridine-3-carboxamide
{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-3-[(3-chlorophenyl)methyl]piperidin-3-yl}methanol
3-(1H-1,2,3-benzotriazol-4-yl)-1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-methylurea
N-[4-(4-methylbenzamido)phenyl]pyrrolidine-3-carboxamide
3-[2-(dimethylamino)ethyl]-8-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[1-(1-{spiro[2.4]heptane-1-carbonyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-amine
5-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]pyrazin-2-ol
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-1H-imidazo[4,5-b]pyridine
1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(2-methylquinolin-6-yl)piperidin-4-ol