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2-[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]-N-[2-(4-fluorophenyl)ethyl]acetamide
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-3-(pyridin-3-yl)propan-1-one
(4aS,8aR)-6-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
7-[(3-methyl-3-phenylpiperidin-1-yl)methyl]-2-(methylsulfanyl)-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
4-(4-phenyl-5-propyl-1H-imidazol-2-yl)-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-[(2E)-2-methylbut-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-5-(1H-indol-1-ylmethyl)-1H-pyrazole-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-2-one
5-(5-ethyl-1,3-oxazol-4-yl)-3-(thiophen-2-yl)-1,2,4-oxadiazole
1-(5-{[(furan-2-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(piperidin-1-yl)propan-2-ol
1-[2-(2-phenylethyl)-1,3-benzoxazole-5-carbonyl]piperidin-4-ol
4-(2-oxoimidazolidine-4-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
4-[6-oxo-3-(pyridin-3-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-1H-pyrazole-3-carboxylic acid
N,N-dimethyl-4-[({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amino)methyl]aniline
1-{3-[3-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidin-4-ol
methyl 1-benzyl-5-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-methyl-2-(3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide
N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
1-(3-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
2,2-dimethylpropyl 2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxylate
1-methyl-N-({5-methyl-2-[3-(propane-2-sulfonamido)phenyl]-1,3-oxazol-4-yl}methyl)cyclohexane-1-carboxamide
4-(5-chloro-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
1-(3-methoxybenzoyl)-4-(3-methyl-1,2-oxazole-5-carbonyl)piperazine
3-(1-methylpiperidin-3-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide
7-(cyclobutylmethyl)-2-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
2-{2-[bis(propan-2-yl)carbamoyl]phenyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1'-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(morpholin-4-yl)butan-1-one
N-(2,2-difluoroethyl)-4-{[(2S)-pyrrolidin-2-ylmethyl]sulfamoyl}benzamide
({5-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
(3S,4S)-1-(2,2-diphenylethyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
4-(1-methyl-1H-imidazol-2-yl)-1-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole
methyl 3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(3-hydroxypropyl)-9-(2-methoxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(4-chloro-2-methylbenzoyl)piperidine
(1s,4s)-4-{4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
3-[4-(1-propylpiperidin-4-yl)piperazin-1-yl]phenol
1-[1-ethyl-5-(2-methoxypyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N,N-dimethyl-2-({2-[4-(propan-2-yl)morpholin-2-yl]acetamido}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)spiro[2.4]heptane-1-carboxamide
N-{1-[(4-fluorophenyl)methyl]-7-[3-(methoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
4-{[4-(5-chlorothiophen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-ethylpyrimidine
9-(5,6-dimethylpyrimidin-4-yl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-chloro-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]pyridine-2-carboxamide
2-{1-azabicyclo[3.2.1]octan-5-yloxy}-N-(pyridin-2-yl)benzamide