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N-[3-(3-methylphenyl)phenyl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-3-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-2-(1H-1,2,4-triazol-3-yl)benzamide
N-(2-{4-[(4-phenylpiperidin-1-yl)methyl]phenoxy}propyl)pyridine-3-carboxamide
9-(2-fluoro-2-phenylacetyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-3-yl}propanamide
1-{3-oxo-3-[4-(pyrimidin-4-yl)piperidin-1-yl]propyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-benzyl-6-(cyclopropylmethoxy)-4-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-1,4-diazepan-2-one
N,N-dimethyl-5-(1,2,3,4-tetrahydroisoquinolin-5-yl)furan-2-carboxamide
4-methoxy-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamide
(2-{[4-(isoquinoline-1-carbonyl)piperazin-1-yl]methyl}phenyl)methanol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
3-methyl-7-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-{2-[4-(trifluoromethyl)phenyl]ethyl}piperidin-4-amine
1-cyclobutanecarbonyl-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
2-(3-methyl-5-{[4-(methylsulfanyl)phenyl]methyl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
N-[(2R,3R)-2-methoxy-1'-[(3-methylthiophen-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
1-(4-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
N-(1-{1-[(3,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-2-carboxamide
ethyl 4-(6-{[4-(methoxycarbonyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-amido)piperidine-1-carboxylate
5-[(3-cyano-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)methyl]-N-methylfuran-2-carboxamide
(1-{[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanamine
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(cyclopropylmethyl)propylamine
5-(3,5-dimethyl-1H-pyrazol-4-yl)-2-methoxypyridine
N-methyl-3-{methyl[(3,4,5-trifluorophenyl)methyl]amino}butanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
8-acetyl-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N,N-diethyl-1-[1-(naphthalen-2-ylmethyl)-7-oxoazepan-4-yl]piperidine-3-carboxamide
2-benzyl-N-(3-hydroxy-3-phenylpropyl)-N-methyl-1,3-thiazole-4-carboxamide
1-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)-1,4-diazepane
4-(3-hydroxy-3-methylbutyl)-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]benzamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[2,6,6-trimethyl-4-oxo-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]naphthalene-1-carboxamide
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-7-(1,3-thiazol-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-2-oxo-N,3-diphenyl-1,8-diazaspiro[4.5]decane-8-carboxamide
N-[(2R,3R)-1'-[2-(cyclohex-1-en-1-yl)acetyl]-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
(1R,2S,6R,7S)-4-[5-(morpholine-4-carbonyl)pyridin-2-yl]-4-azatricyclo[5.2.2.02,6]undecane
2-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[2-(piperidin-1-yl)ethyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)(pyridin-4-ylmethyl)amine
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
2-(4-fluorophenyl)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
9-(4-hydroxybenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-4-{[(2,5-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
N-(1-benzothiophen-2-ylmethyl)-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one