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4-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]pyridin-2-amine
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[1-(4-methoxyphenyl)ethyl]-N-methylpropanamide
(3R,4R)-1-(6,8-dimethylquinolin-4-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
(3aS,7aR)-2-(1H-1,2,3-benzotriazole-5-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(5-fluoro-2-methylphenyl)ethan-1-one
1-cyclopropyl-5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]piperidin-2-one
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[2-(furan-2-yl)ethyl]amine
N-{[(2S,4S)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-fluoropyrrolidin-2-yl]methyl}propanamide
N-(2H-1,3-benzodioxol-5-yl)-7-(oxolane-2-amido)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[3-(1H-indol-2-yl)phenyl]-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]piperidin-4-amine
1-{2-[2-(2-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
2-(2-{[2-(dimethyl-1,3-thiazol-2-yl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
6-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
3-methyl-7-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-{1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]piperidin-4-yl}pyridin-2-amine
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(pyridine-4-carbonyl)-1,4-diazepan-2-one
4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]-N-[2-(2-methoxyphenyl)ethyl]benzamide
(2-{2-[1-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}propanamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
N-(2,3-dihydro-1H-inden-2-yl)-1-(6-ethoxy-4-methylquinazolin-2-yl)piperidin-4-amine
2-methoxy-4-{3-methyl-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
3-(hydroxymethyl)-N-(isoquinolin-5-yl)morpholine-4-carboxamide
1-[(3-fluorophenyl)methyl]-6-oxo-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
2-(4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazin-1-yl)benzonitrile
5-(furan-2-ylmethyl)-5-{3-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}pyrrolidin-2-one
3-methyl-7-[4-(2-methylpropyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(1S,5R)-N-cyclopentyl-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(2,4,6-trifluorophenyl)acetamide
1-[1-(3-cyano-6-methylpyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
5-[4-(3-methylphenoxy)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
1-(2,4-dimethoxyphenyl)-3-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}urea
{[4-ethyl-5-(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
3-[(2,5-dimethylphenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]-2-(2-methoxyphenoxy)acetamide
1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-[(1S,5R)-3-[2-(benzyloxy)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
6-methyl-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-(pyridin-3-yl)pyrimidin-4-amine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
4-(pyridin-3-ylmethyl)-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
N-({7-[4-(dimethylamino)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(pyrazin-2-yl)ethan-1-one
1-(furan-2-ylmethyl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]piperidin-4-amine
N-[2-(diethylamino)ethyl]-N-ethyl-2-(thiomorpholin-4-yl)-6-(thiophen-2-yl)pyridine-3-carboxamide
1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-3-(3-methoxyphenyl)propan-1-one
4-(4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)quinazoline
3-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-indazole
N-[(3,5-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-2-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-[(1-benzylpyrrolidin-3-yl)methyl]-2,4-difluorobenzamide