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1-(4-methoxyphenyl)-6,6-dimethyl-4-(2-methylbutanoyl)piperazin-2-one
2-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-1H-imidazole
6-[(3,4-dimethylphenyl)methyl]-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-({7-[3-(prop-2-en-1-yloxy)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
3-(2,5-difluorobenzoyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
1-[(3,4-dimethylphenyl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
1-[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-[(2-methylphenyl)methyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
4-{5-[(2,3-difluoro-6-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-1H-pyrazole
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(thiophen-3-yl)propanamide
1-(azepan-1-yl)-3-[3-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4R)-4-(4-{2-[(3-methoxyphenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-cyclopropyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(pyridin-4-ylmethyl)acetamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
2-[1-(1,7-dimethyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]-6-methyl-1H-1,3-benzodiazole
(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}morpholin-2-yl)methanamine
2-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(2-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}quinolin-6-yl)acetamide
3-({[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]amino}methyl)pyrrolidin-3-ol
1-{[5-(3-fluorophenyl)-1,2,4-triazin-3-yl]amino}butan-2-ol
7-(1H-inden-2-yl)-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1-(1H-pyrazol-1-ylmethyl)cyclopropane-1-carboxamide
4-[(5-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
N-benzyl[(3-oxo-1,3-dihydro-2-benzofuran-5-yl)amino]sulfonamide
1-{4-[(3,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-3-phenylpropan-1-ol
2-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
benzyl 4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxylate
1-(3-methoxy-4-methylphenyl)-3-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]urea
3-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-(1-benzylpyrrolidin-3-yl)propanamide
2-({6-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
(4aR,6R,8aS)-2-benzoyl-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
methyl 9-[2-(2-fluorophenyl)ethoxy]-7-oxo-3-(4-oxopentanoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(pyrrolidin-3-yl)piperazine
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(2-methylbutyl)acetamide
1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
N-(2,4-difluorophenyl)-4-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}benzamide
1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
2-(2-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)-N-ethylacetamide
4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[4-(pyridin-4-yl)piperidin-1-yl]butan-1-one
1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-2-(2-methyl-1H-indol-3-yl)ethan-1-one
(3aS,6aR)-5-[(2-methyl-1-benzothiophen-3-yl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepan-5-one
1-[3-(3-ethylphenoxy)azetidin-1-yl]-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
1-(5-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-(furan-2-ylmethyl)pyrimidin-2-amine