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{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-[(4-hydroxy-3-methylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-butyl-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1,3-benzoxazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-4-(1H-pyrazol-1-yl)benzamide
8-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
4,4,4-trifluoro-3-[2-(4-propanoylphenoxy)acetamido]butanoic acid
methyl 8-{[4-(2-hydroxyethoxy)phenyl]methyl}-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
5-methyl-1-(3-{2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}phenyl)-1H-1,2,3,4-tetrazole
N-[1-(4-chlorophenyl)ethyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
5-(azepane-1-carbonyl)-N-[(3-chlorophenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-cyclopropyl-8-[2-(4-ethylpiperazin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-cyclopropyl-5-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazole
N-[2-(azepan-1-yl)ethyl]-2-(dimethylamino)-2-(4-methylphenyl)acetamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(pyridin-3-yloxy)propyl]benzamide
(5S,9aS,9bS)-5-(4-methoxy-2,3-dimethylphenyl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
6-[(diethylamino)methyl]-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
methyl 4-{[methyl(1,2,3,4-tetrahydronaphthalen-1-yl)amino]methyl}-1H-pyrazole-3-carboxylate
2-[(3aS,6aR)-3-[(2-methoxyphenyl)methyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]-4,6-dimethylpyridine-3-carbonitrile
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-(pyridin-4-yl)propan-1-one
N-(3-methoxypropyl)-6-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(3R,9aR)-8-(3-methoxybenzoyl)-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(4-chlorophenyl)methyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(4aR,7aS)-1-(2-hydroxyethyl)-4-{[4-(methylsulfanyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
1-ethyl-N-[(4-fluorophenyl)methyl]-N-(2-methylpropyl)-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperidin-4-yl}-1,3-oxazolidin-2-one
(1s,4s)-4-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)cyclohexan-1-ol
2-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-1H-indole
1-{[5-(3-phenylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,4-diazepan-5-one
{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amine
methyl 4-[2-amino-3-cyano-6-(1,3-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
2-benzyl-8-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-(1-methylpiperidin-4-yl)-4-(methylsulfanyl)-N-(pyridin-4-ylmethyl)benzamide
8-{[2-(furan-2-yl)phenyl]methyl}-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[(2-methylphenyl)(pyridin-4-yl)methyl]piperidine-4-carboxamide
2-({7-chloro-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N,5-dimethyl-1-propyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(4-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
1-(cyclopropylmethyl)-4-(2,4-dimethoxybenzoyl)-2-(propan-2-yl)-1,4-diazepane
2,6-difluoro-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
1-[(3-ethoxy-4-methoxyphenyl)methyl]-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
6-(morpholin-4-yl)-N4-(pyridin-4-ylmethyl)pyrimidine-2,4-diamine
3-phenyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazine
2-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-5-(1-methyl-1H-pyrazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(3,5-dimethylfuran-2-carbonyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
1-[3-({[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol