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1-[(4-chlorophenyl)methyl]-N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
(2S)-2-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}propanamide
6-[4-(morpholin-4-yl)benzoyl]-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
7-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[1-(thiophen-2-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
(2S,4R)-N,N-dimethyl-4-[(4-methylpyrimidin-2-yl)sulfanyl]-1-[(4-phenylphenyl)methyl]pyrrolidine-2-carboxamide
3-chloro-N-ethyl-2-fluoro-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-{1-[(3-methoxyphenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[4-(benzyloxy)butyl]benzamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-N-ethyl-4-(3-methyloxetane-3-amido)pyrrolidine-2-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperazine
3-{[(dimethylcarbamoyl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
ethyl 3-[(2-fluorophenyl)methyl]-1-(5-methyl-1H-pyrazole-3-carbonyl)piperidine-3-carboxylate
3-(1H-indol-3-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}propanamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
3-(2-chlorophenyl)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
3-{1-[(3-fluorophenyl)methyl]-1H-pyrazol-4-yl}-1-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
1-[2-(2-phenylpyrrolidine-1-carbonyl)phenyl]-1H-1,2,4-triazole
ethyl 4-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]piperidine-1-carboxylate
2-(2-methoxyethyl)-5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}pyrimidine
N-(2-methoxyethyl)-N-methyl-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(quinoline-4-carbonyl)pyrrolidin-3-yl]methanol
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}propanamide
9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-3-(thiophene-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl})amine
N4-[(1-phenylpyrrolidin-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
8-chloro-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]quinoline
1-(3-phenyl-1,2-oxazole-5-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
1-[(3-methoxyphenyl)methyl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazin-2-one
N-ethyl-N-(2-hydroxyethyl)-2-[3-(4-methoxyphenyl)-1-(3-methylbutyl)-2,5-dioxopyrrolidin-3-yl]acetamide
1-(2,4-dimethylphenyl)-3-[3-(methylsulfanyl)propyl]urea
2,3-dichloro-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-3-propanamidobenzamide
N-{[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-2-carboxamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(methylsulfanyl)ethyl]pyridin-2-amine
3-[(3-fluorophenyl)methyl]-N-[(1R)-1-(4-methoxyphenyl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
3-{[(2R,3R)-3-(3-fluorobenzamido)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]carbonyl}pyridin-1-ium-1-olate
methyl 4-({4-[4-methyl-2,5-dioxo-1-(thiophen-3-ylmethyl)imidazolidin-4-yl]piperidin-1-yl}methyl)benzoate
6-{[2-(dimethylamino)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-en-8-yl]methyl}pyridine-2-carboxylic acid
2-butyl-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidin-3-ol
1-methyl-N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,3-benzodiazole-5-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-5-methyl-1,3-oxazole-4-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]pyrimidin-2-amine
3-[(3-ethoxyphenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-(4-methylphenyl)-3-oxo-3-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}propanamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
6-[(3-fluorophenyl)methoxy]-4-(2-methyl-1,3-thiazole-4-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
2,2,3-trimethyl-N-[(1-methylpyrrolidin-3-yl)methyl]but-3-enamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-4-(piperidin-1-yl)butanamide