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3-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-4-(2-methylpropyl)piperazin-2-one
3-benzyl-1-(3-methoxypropyl)-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,5S)-5-[(pyridin-2-ylmethyl)carbamoyl]-1-(1H-pyrrole-2-carbonyl)piperidine-3-carboxylic acid
N-(1-cyclopropylethyl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
2-chloro-6-methoxy-4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{3-[(5-methylpyridin-2-yl)amino]propyl}acetamide
(4aR,8aS)-N,N-dimethyl-1-(3-methylbenzoyl)-decahydro-1,6-naphthyridine-6-sulfonamide
6,8-difluoro-4-{4-[1-(morpholin-4-yl)ethyl]phenyl}quinoline
ethyl 1-[1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperidine-3-carboxylate
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-2-{[(2-methylphenyl)methyl]sulfanyl}acetamide
N-[2-(4-hydroxyphenyl)ethyl]-3-methyl-5-propyl-1-benzofuran-2-carboxamide
(2S,4S)-1-[(2E)-but-2-en-1-yl]-4-[3-(dimethylamino)benzamido]-N-ethylpyrrolidine-2-carboxamide
2-[4-(4-acetylphenyl)piperazin-1-yl]-N-methyl-N-(1-methylpiperidin-4-yl)-6-(4-methylthiophen-2-yl)pyridine-3-carboxamide
[1-(2,5-dimethoxyphenyl)ethyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
4-(5-hydroxypyrazine-2-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
3-[2-(azepan-1-yl)-2-oxoethyl]-4-(thiophen-2-ylmethyl)piperazin-2-one
N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-propanoylpiperidine-3-carboxamide
(2S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
3-[3-cyclopropyl-1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl]-1-phenylpropan-1-one
5-(2-methylpropyl)-1'-(6-methylpyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-benzyl-2-{2-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
2-{[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}-6-fluoroquinolin-4-ol
N-methyl-N-(naphthalen-1-ylmethyl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{2-[(6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)formamido]ethyl}acetamide
[1-(1-benzothiophene-2-sulfonyl)-3-benzylpiperidin-3-yl]methanol
methyl 6-[(3S,4R)-3-acetamido-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]pyrimidine-4-carboxylate
4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(methylsulfanyl)propanamide
5-oxo-1-(propan-2-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidine-3-carboxamide
4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine-1-sulfonamide
4-{6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}-1,4-diazepane-1-carbaldehyde
1-methyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}phthalazine
1-ethyl-3-(2-methylpropyl)-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-5-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
1-methyl-N-[3-(4-methylbenzenesulfonamido)propyl]-1H-indole-6-carboxamide
N,N,2-trimethyl-7-{2-methylthieno[3,2-d]pyrimidin-4-yl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-(4-methoxyphenyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1,2,4-oxadiazole
N-[(4-fluorophenyl)methyl]-3-[1-(6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-4-yl]propanamide
6-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)(phenyl)methanol
4-[4-(3-hydroxyphenyl)piperidin-1-yl]pyrimidine-5-carboxylic acid
2-{4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazin-1-yl}pyrazine
1-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
6-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)pyridine-2-carboxylic acid
1-(6-hydroxypyridine-3-carbonyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-[2-(4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperazine
N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-methyl-1-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}urea
N-[(3-ethoxyphenyl)methyl]-N-(prop-2-en-1-yl)oxane-4-carboxamide