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1-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
2-({3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)-4-methoxyphenol
6-(cyclopropylamino)-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
5-(furan-3-carbonyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(3-methoxyphenyl)-5-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1,3-thiazol-2-amine
N-(3,5-dimethoxyphenyl)-3-{[(2,5-dimethylphenyl)methyl]amino}-5-(dimethylsulfamoyl)benzamide
2-[3-(3-fluorophenoxymethyl)-5-(2-methanesulfonamidoethyl)-1H-1,2,4-triazol-1-yl]acetic acid
ethyl 5-({[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidin-2-yl]formamido}methyl)furan-2-carboxylate
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
methyl 5-[(2R,3R)-2-ethoxy-3-(pyridine-3-amido)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-5-oxopentanoate
N-(cyclopropylmethyl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
6-methyl-3-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
methyl 3-(2-methoxybenzamido)-5-({2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamido}methyl)benzoate
N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
ethyl 1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-phenylethyl)piperidine-3-carboxylate
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-(4-fluoro-2-methylphenyl)-3-[1-(1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
N-(1-{7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylbenzamide
4-ethenyl-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
1-ethyl-8-[4-(4-hydroxyphenyl)butan-2-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
N-(8-chloroquinolin-5-yl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
N-(3,4-dimethylphenyl)-2-{[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]amino}acetamide
2-(2,5-dimethoxyphenyl)-N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}acetamide
5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)-5-[1-(3-methylpentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[2-hydroxy-3-(piperazin-1-yl)propyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-cyanobenzene-1-sulfonamide
1-{4-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(thiophen-3-yl)ethan-1-one
(4aS,8aR)-6-(3,5-difluorobenzoyl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
1-methyl-5-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(4aR,7aS)-1-(1H-imidazol-4-ylmethyl)-4-[3-(pyridin-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-1-{4-[2-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}propan-1-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(3-methylbutyl)piperidine-3-carboxamide
2-{3-[({[4-(methylsulfanyl)phenyl]methyl}(propyl)amino)methyl]phenoxy}ethan-1-ol
3-(1H-indol-3-yl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]propanamide
ethyl 4-(3-phenylpropyl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylate
2-{2-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-1-cyclopentylpiperazin-2-yl)ethan-1-ol
(4aS,7aR)-1-(3-phenylpropanoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}-N-[(3S)-pyrrolidin-3-yl]benzamide
[1-(2-methoxyphenyl)propan-2-yl]({1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-imidazole