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1-methyl-6-oxo-N-[1-(thian-4-yl)piperidin-4-yl]-1,6-dihydropyridazine-3-carboxamide
1-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(2-chlorophenyl)ethan-1-one
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(1H-imidazol-1-yl)propyl]propanamide
N-({3-methyl-7-[4-(trifluoromethyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
2-amino-4-(3-chloro-4-hydroxyphenyl)-6-(5-methylpyridin-2-yl)pyridine-3-carbonitrile
N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-ethyl-N-(4-hydroxybutyl)-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)propanamide
2,5-difluoro-N-({5-methyl-2-[2-(3-phenoxypropanamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
N-(2H-1,3-benzodioxol-5-yl)-6-(cyclopent-1-ene-1-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-methyl-N-({8-[(2,3,6-trifluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-thiazole-4-carboxamide
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-{4-[(2E)-3-phenylprop-2-en-1-yl]morpholin-3-yl}acetamide
N-[(2R,3R)-2-methoxy-1'-(3-phenoxypropanoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
2-{5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-(1H-imidazol-4-ylmethyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
2-({4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
N-[(2S,4R,6S)-2-[2-(benzyloxy)phenyl]-6-ethyloxan-4-yl]acetamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}[(6-methylpyridin-2-yl)methyl]amine
1-{4-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]phenyl}ethan-1-one
4-({[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
1-methyl-2-phenyl-4-(1,3-thiazol-4-ylmethyl)piperazine
{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}[(2,3,5-trimethyl-1H-indol-7-yl)methyl]amine
1-(3-methylbut-2-en-1-yl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-benzyl-3-[4-(3-cyanopyrazin-2-yl)piperazin-1-yl]-N-ethylpropanamide
6-(piperidin-3-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyrimidin-4-amine
(1H-indol-6-ylmethyl)(methyl)[2-(morpholin-4-yl)ethyl]amine
4-(4-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
9-methoxy-3-(2-methylbutyl)-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-[2-(4-methoxyphenyl)ethyl]-4-(4-methyl-1,4-diazepan-1-yl)pyridine-2-carboxamide
N-{[8-(4-fluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}isoquinoline-3-carboxamide
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
ethyl 2-(1-{[3-(methylsulfanyl)phenyl]carbamoyl}piperidin-2-yl)acetate
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
1-(2,3-dimethylphenyl)-4-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperazine
1-{3-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-oxopropyl}pyrrolidin-2-one
N-(2-phenylpropyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methylpiperidine-2-carboxamide
N-{4-[({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}carbamoyl)methyl]phenyl}butanamide
4-{pyrazolo[1,5-a]pyrimidin-3-yl}phenol
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[(1r,4r)-4-hydroxycyclohexyl]-1H-1,3-benzodiazole-5-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-(1,3-benzothiazol-2-ylmethyl)acetamide
methyl 3-ethyl-2-[2-(trifluoromethyl)morpholin-4-yl]-3H-imidazo[4,5-b]pyridine-6-carboxylate
1-[(2,4-difluorophenyl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
3-(2-phenylethyl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
N-(2-phenylethyl)-6-[2-(3,4,5-trimethoxyphenyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
5-(2-methoxyacetamido)-N-(3-methoxypropyl)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide