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N-(5-{[3-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]methyl}thiophen-2-yl)acetamide
3-[5-(2-cyclopentylethyl)-4-phenyl-1H-imidazol-1-yl]propanamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-(4-ethylpiperazin-1-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,3-dihydro-1H-indene-2-carboxamide
2-{[5-(2-chlorophenyl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(4aR,7aS)-1-acetyl-4-[(3,5-dichlorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(thiophen-3-yl)ethan-1-one
1-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-3-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)urea
N-(4-methoxy-2-methylphenyl)-3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]propanamide
5-(oxolan-2-yl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]thiophene-2-carboxamide
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-1-[(4-methoxy-3-methylphenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyrrolidine-2-carboxamide
N,2-dimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
2-({[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)ethan-1-ol
3-methyl-7-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-N-benzylpyrimidin-2-amine
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-(2,2,2-trifluoroethyl)propanamide
1-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-4-phenyl-1,2,3,6-tetrahydropyridine
N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-3-phenylpropanamide
ethyl 1-(5,8-dimethoxy-3-{[(2-phenylethyl)amino]methyl}quinolin-2-yl)piperidine-4-carboxylate
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
1-(4-chlorophenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)cyclopropane-1-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-N-(2-methoxyethyl)-2-methylthieno[2,3-d]pyrimidin-4-amine
2-{1-[(3,4-difluorophenyl)methyl]-4-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
6-[(2-ethoxyphenyl)methyl]-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]urea
(3R,4R)-4-(azepan-1-yl)-1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-ol
2-(4-methoxyphenyl)-6-(pyrrolidine-1-carbonyl)pyrazine
2-{[(1R)-1-(4-fluorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-methyl-2-[2-(oxan-2-ylmethyl)phenoxy]acetamide
N-[phenyl(pyridin-4-yl)methyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-cyclohexyl-N3-[2-(3,4-dimethoxyphenyl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{1-[1-(carbamoylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
1-(2-{[(pyridin-3-ylmethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-(4-{[(3-methoxyphenyl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(4aR,7aS)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(2-phenylpropyl)propanamide
7-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{4-[2-(piperazin-1-ylmethyl)phenyl]phenyl}acetamide
(3R,5S)-N-[3-(dimethylamino)propyl]-1-(pyridin-4-ylmethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
methyl 3-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2-hydroxyethyl)-1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-phenyl-1H-pyrazole-3-carboxamide
2-(3-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}phenoxy)acetamide
(3R,4R)-4-ethyl-1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidine-3,4-diol
2-{1-[(6-methoxypyridin-3-yl)methyl]pyrrolidin-2-yl}-1-methyl-1H-1,3-benzodiazole
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-methyl-1-[2-(morpholin-4-ylmethyl)phenyl]-3-[(5-propyl-1H-pyrazol-3-yl)methyl]urea
5-ethyl-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-hydroxy-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide