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1-[(4-ethylphenyl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[2-(1H-pyrazol-1-yl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
N-(3,5-dimethoxyphenyl)-2-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]acetamide
N-{7-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1-ethyl-2-(pyridin-3-yl)-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
(1S,5R)-6-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
4-(cyclopropylmethyl)-1-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-3-(propan-2-yl)-1,4-diazepan-5-one
2-(methylsulfanyl)-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyridine
1-(3-{4-[2-(3-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)ethyl]piperazine-1-carbonyl}phenyl)pyrrolidin-2-one
N-methyl-N-{3-oxo-3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}methanesulfonamide
2-amino-7-(3-chloro-4-ethoxybenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methylpentanamide
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-1-cyclopropyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
methyl 4-(4-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)amino]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-7-fluoro-3-methyl-1-benzofuran-2-carboxamide
4-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-N-(oxan-3-ylmethyl)pyrimidin-2-amine
methyl 1-{[1-(cyclobutylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}piperidine-4-carboxylate
(2E)-1-[4-(4-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
1-(1,2-oxazolidin-2-yl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
(3S,4S)-1-(ethanesulfonyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-(carbamoylmethyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxamide
N-(2-{5-methyl-4-[(2-phenylpropanamido)methyl]-1,3-oxazol-2-yl}phenyl)pyridine-3-carboxamide
N-[(2R,3R)-1'-benzoyl-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
3-{2-oxo-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethyl}-2,3-dihydro-1H-isoindol-1-one
2-amino-8-[4-(4-chlorophenyl)butanoyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[(1-methylpiperidin-3-yl)methyl]-4-oxo-4-phenylbutanamide
4,4,4-trifluoro-N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}butanamide
7-(2-methylphenyl)-4-(2-propoxyethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
1-(3-methylpyridin-2-yl)-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-1H-indole
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
methyl 3-(oxolane-3-amido)-5-[(pentan-3-yl)amino]-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridin-3-ol
6-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carbonitrile
5-{3-[(2S)-4-methyl-2-phenylpiperazin-1-yl]-3-oxopropyl}-5-(thiophen-2-ylmethyl)pyrrolidin-2-one
[1-(cyclohexylmethyl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol
1-[1'-(5-hydroxypyrazine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
2-[(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)amino]acetic acid
4-(1-benzothiophen-7-yl)-6-methylpyrimidin-2-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-methoxy-2-(thiophen-2-yl)ethyl]amine
3-[2-(4-fluorophenyl)piperidin-1-yl]-N-(furan-2-ylmethyl)propanamide
4-(ethanesulfonyl)-2-[(3-fluorophenyl)methyl]morpholine
3-(3-methoxyphenyl)-N-methyl-N-[1-(pyridin-3-yl)ethyl]benzamide
(1S,5R)-6-methyl-3-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one