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4-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]-1-phenylpiperazin-2-one
4-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl]benzonitrile
2-methoxy-N-[(2R,3R)-2-methoxy-1'-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
(5S,9aS,9bS)-5-(2-chloro-4-fluorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
[(1-cyclohexylpiperidin-3-yl)methyl]({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(pyridin-3-ylmethyl)amine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-benzoxepine-4-carboxamide
(4aR,7aS)-1-methanesulfonyl-4-(2-methyl-1,3-thiazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2H-1,3-benzodioxol-5-yl)-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)acetamide
N-methyl-N-[2-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]methanesulfonamide
5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)-5-[1-(4-oxopentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
3-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-1,5,6-trimethyl-1,2-dihydropyridin-2-one
2-methoxyethyl 3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxylate
2-methoxy-1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-2-phenylethan-1-one
3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-1-(thiomorpholin-4-yl)propan-1-one
3-(2H-1,3-benzodioxol-5-yl)-N-ethyl-3-phenyl-N-(pyridin-4-ylmethyl)propanamide
2-(3-cyclohexyl-1,2,4-oxadiazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-amino-6-{4-[4-(ethylamino)pyrimidin-2-yl]piperazin-1-yl}-3,4-dihydropyrimidin-4-one
N-[(2R,3R)-2-ethoxy-1'-(4-fluorobenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
N-(2,3-dihydro-1H-inden-1-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(quinolin-3-ylmethyl)benzamide
7-(cyclopropylmethyl)-2-(3-phenoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[3-(pyrimidin-2-yloxy)phenyl]methyl}amine
1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]-2-(thiophen-2-yl)ethan-1-one
N-{[1-(2,2-dimethylpropyl)piperidin-4-yl]methyl}-3-hydroxybenzamide
4-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}azetidin-3-yl)morpholine
N-(1-benzothiophen-2-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
3-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carbonyl]-1H-indazole
1-[2-(dimethylamino)ethyl]-6-oxo-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)piperidine-3-carboxamide
N5-benzyl-N5,N6-dimethyl-N6-[1-(pyrimidin-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carbonyl]pyridine
1-{4-[4-(2-methylphenoxy)piperidin-1-yl]-4-oxobutyl}piperidin-2-one
4-(2,1,3-benzothiadiazol-4-yl)-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
N-cyclopentyl-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-[1'-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-(2-methoxyethyl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1,3-benzoxazole-6-carboxamide
1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-4-propylpiperazine
(3S,4S)-1-[1-(2-chlorophenyl)piperidin-4-yl]-4-(morpholin-4-yl)pyrrolidin-3-ol
2-[3-(4-fluorophenyl)-4-methyl-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
N-[(4-fluorophenyl)methyl]-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
6-{[(3R,4S)-4-cyclopropyl-1-(oxane-4-carbonyl)pyrrolidin-3-yl]amino}pyrazine-2-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]piperazine
2-cyclobutyl-N-(3-hydroxypropyl)-1-methyl-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
7-[(4-fluorophenyl)methyl]-2-[(2-methoxypyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decane
1-[3-(difluoromethoxy)benzoyl]-4-(4-fluorophenyl)-1,4-diazepane
N-{[8-(4-fluorobenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2,4-dimethoxybenzamide