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5-[1-(1H-pyrazol-1-yl)ethyl]-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
2-methyl-4-oxo-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
1-[3-({[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
5-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1-[(2-methoxyphenyl)methyl]-N-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[methyl(pyridin-3-ylmethyl)amino]-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
3-ethyl-5-{[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]methyl}-4,5-dihydro-1,2-oxazole
3-chloro-N-cyclopentyl-4-{[1-(1-ethylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-methylbenzamide
(3aR,6aR)-2-cyclopentyl-5-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
8-cyclopentyl-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[4-(propan-2-yl)phenyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-3-amine
(1S,5R)-3-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(cyclopropylmethyl)-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aR,8aS)-6-[(2,3-dimethoxyphenyl)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-1-ethyl-3-methyl-1H-pyrazole-4-carboxamide
(2-{2-[1-(1H-indazole-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-(4-hydroxypiperidin-1-yl)-2-[4-(4-{[1-(naphthalen-1-yl)ethyl]amino}piperidin-1-yl)phenyl]ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3,3-dimethylbutanoyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3S,4R)-1-[(1-benzyl-1H-imidazol-5-yl)methyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
3-(2-fluorophenyl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
2,3,6-trifluoro-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)benzamide
N-(1-{1-[2-(2-methylphenyl)benzoyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
3-{1-[1-(2-aminoacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-chlorophenyl)urea
2-(2,3-difluorophenoxymethyl)-N-(prop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(5-methyl-1H-pyrazol-1-yl)acetamide
4-benzyl-3-ethyl-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-1,4-diazepan-5-one
(1S,5R)-3-(pyrimidin-2-yl)-6-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-methylpyridine-3-carboxylic acid
N-ethyl-2-[(isoquinolin-5-yloxy)methyl]-N-(oxan-4-yl)-1,3-oxazole-4-carboxamide
1-ethyl-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)piperidin-4-amine
4-[1-cyclohexyl-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazol-3-yl]pyridine
N,8-dimethyl-3-({methyl[2-(morpholin-4-yl)ethyl]amino}methyl)-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1H-indole-2-carbonyl)-2,7-diazaspiro[4.5]decane
(3S)-3-benzyl-4-[(4-methoxy-2,5-dimethylphenyl)methyl]piperazin-2-one
3-({[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
5-(3-fluorophenyl)-4-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-2-(trifluoromethyl)pyrimidine
2-fluoro-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(3-phenylpropyl)propanamide
1-(3-phenylpropyl)-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
N-(furan-3-ylmethyl)-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N,N-bis(prop-2-en-1-yl)acetamide
6-(2-methoxyphenyl)-N-methyl-N-(thiophen-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{1-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}pyridine
N-(2-hydroxyethyl)-1-methyl-N-[(3-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[4-(pyrrolidin-1-ylmethyl)phenyl]-1H-indazole
6-cyclopentyl-3-{[(5-ethyl-2-methylpyrimidin-4-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one