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4-[2-(oxolan-3-yl)ethyl]-1-(2-phenylphenyl)piperazin-2-one
N-(2,2,2-trifluoroethyl)-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
[(1,3-dimethylpyrrolidin-3-yl)methyl][(5-fluoro-1-methyl-1H-indol-2-yl)methyl]methylamine
(3R,5S)-N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
methyl (2S,4R)-1-[(3-chlorophenyl)methyl]-4-(2,2-diphenylacetamido)pyrrolidine-2-carboxylate
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[4-(methylsulfanyl)phenyl]acetamide
1-ethyl-4-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)pyrrolidin-2-one
3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-2-oxopentanamide
2-methyl-1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-1,4-diazepan-5-one
2-{3-[4-(3-methylphenoxy)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
N-(4-cyano-2-fluorophenyl)-4-(4-methyl-1H-pyrazol-3-yl)piperidine-1-carboxamide
1-{[4-(methylsulfanyl)phenyl]methyl}-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
2-(4-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
3-ethyl-4-[2-(4-fluorophenoxy)acetyl]-3-methylpiperazin-2-one
1-{2,8-diazaspiro[4.5]decane-3-carbonyl}-4-phenylpiperidine-4-carbonitrile
N-(2-methanesulfonamidoethyl)-2-(4-propanoylphenoxy)acetamide
4-ethyl-3-(piperidin-4-ylmethyl)-1-[3-(1H-pyrazol-1-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-methyl-7-(1-phenylcyclopropanecarbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(furan-3-carbonyl)-1,4-diazepane
methyl 2-{4-[(1-ethyl-1H-pyrazol-3-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
N-(1-benzylpiperidin-4-yl)-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-{[(4-methyl-5-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]methyl}pyridine
(3aR,6aS)-2-(3-methoxy-5-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-chloro-5-acetamido-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
1-cyclobutanecarbonyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-4-carboxamide
1-[4-(aminomethyl)piperidin-1-yl]-2-{[(2-chlorophenyl)methyl]sulfanyl}ethan-1-one
4-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2,3-dihydro-1H-imidazol-2-one
{2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}urea
3-(4-{[4-(3,4-dimethylphenoxy)phenyl]methyl}piperazin-1-yl)propanamide
2-{3-cyclopentyl-5-[2-(ethylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-{2-[(2-phenoxyethyl)amino]ethyl}-1-(3-phenylpropyl)pyrrolidin-2-one
6-{[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxyethan-1-one
N,N-dimethyl-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}aniline
2-(4-chloro-2-methylphenoxy)-N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}propanamide
2-{[(4-hydroxy-5,8-dimethylquinolin-2-yl)methyl]amino}-1-(pyrrolidin-1-yl)ethan-1-one
3-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
(3S,4R)-1-{[3-(2-aminoethyl)phenyl]methyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-(1-ethyl-5-oxopyrrolidine-3-carbonyl)-1-[(4-fluorophenyl)methyl]piperazin-2-one
9-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
N-(1-{4-[(2,3-dihydro-1H-inden-2-yl)carbamoyl]phenyl}-1H-pyrazol-4-yl)-2,4-dimethylbenzamide
3-methoxy-N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
2-(3-methylfuran-2-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
2-[3-({3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
(4aS,8aR)-1-(2-methylpropyl)-6-[2-(4-oxo-1,4-dihydropyridin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-[methyl({[1-(propan-2-yl)-1H-imidazol-2-yl]methyl})amino]-1-phenylethan-1-ol
N-({8-[2-(4-chlorophenyl)acetyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide