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4-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-1-(3-chlorophenyl)piperazin-2-one
N-(adamantan-1-yl)-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
6-methyl-5-(2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-9-methyl-9H-carbazole-3-carboxamide
methyl 1-(3-methylbutoxy)-2-oxo-8-(2-phenylethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-(cyclohexylmethyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
6-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-methyl-1-(naphthalen-1-ylmethyl)-N-(oxan-4-yl)-1H-1,2,3-triazole-4-carboxamide
3-phenyl-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]propanamide
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-(3-methylthiophene-2-carbonyl)piperidine
1-methyl-3-[1-(5-oxopyrrolidine-3-carbonyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,4-diazepan-2-one
4-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-2,6-dimethoxyphenol
methyl 3-{[(4-methyl-1H-imidazol-2-yl)formamido]methyl}-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
2-ethyl-8-[(4-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-methyl-N-(1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
2-[(8-chloroquinolin-2-yl)formamido]-N-methylpentanamide
3-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}phenol
2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1,9-dimethyl-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4,4,4-trifluoro-N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
N-methyl-N-{2-[(4,4,4-trifluorobutan-2-yl)amino]ethyl}methanesulfonamide
4-methyl-1-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pentane-1,2-dione
3-(2-fluoro-4-methoxyphenyl)-1-[2-phenyl-2-(piperidin-1-yl)ethyl]urea
2-{1-[(4-fluorophenyl)methyl]-5-{8-methylimidazo[1,2-a]pyridin-2-yl}-1H-1,2,4-triazol-3-yl}acetamide
(2S,4R)-4-[(adamantan-2-yl)amino]-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
dimethyl({4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]butan-2-yl})amine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylpropanamide
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
(4aR,7aS)-1-(pyrimidin-2-yl)-4-(4,4,4-trifluorobutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({1-[2-(diethylamino)acetyl]piperidin-3-yl}methyl)-4-fluorobenzamide
N-({8-[2-(trifluoromethyl)benzoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide
2-[4-(2-methoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
5-ethyl-1'-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(propan-2-yl)piperidine-3-carboxamide
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-3-(1-methylpiperidin-4-yl)propanamide
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
(4aS,7aR)-1-(2-methoxy-4-methylbenzoyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-methyl-3-phenyl-1-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]piperidine
1-(azepan-1-yl)-3-[4-chloro-2-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-(2-phenylethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-(quinolin-6-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
5-{3-[3-(2-chlorophenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-one
1-[(4-chlorophenyl)methyl]-N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
methyl 2-{[5-(4-fluorophenyl)-4-[1-(3-methylbenzoyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
2-{5-methyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]benzamide
ethyl 4-(4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanoyl)piperazine-1-carboxylate