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4-(hydroxymethyl)-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidin-4-ol
2-[({5-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
8-(4-methoxy-2-methylbenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-(pyridin-3-ylmethyl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-benzyl-2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxyethyl)acetamide
(1S,7R)-4-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-phenylcyclohexane-1-carboxamide
3-[(2R,3R,6R)-5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(2S,4R)-1-[2-(3-cyclopropanecarbonyl-1H-indol-1-yl)acetyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
2,3-dimethyl-6-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoxaline
(4-fluoro-3-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)methanamine
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
4-methyl-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]pyrimidine-5-carboxamide
methyl 5-{[(3,5-difluorophenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2,3-dihydro-1-benzofuran-7-yl)-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridine
[3-(cyclopropylmethyl)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperidin-3-yl]methanol
N-methyl-1-phenylmethanesulfonyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
2-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-2-yl}acetic acid
1-[(4,5-dimethylfuran-2-yl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-ethyl-N-{[2-(trifluoromethoxy)phenyl]methyl}pyrimidine-5-carboxamide
3-[(2-chlorophenyl)methyl]-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine
1-ethyl-1-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-3-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]urea
methyl (2S,4R)-1-[(3-methoxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
1-[(1-acetylpiperidin-3-yl)methyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
1-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-5-phenylpentan-1-one
methyl 1-{2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-2-carboxylate
2-[(1-ethyl-1H-imidazol-2-yl)methyl]-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
3-[2-(4-cyclohexylpiperazin-1-yl)-2-oxoethyl]-4-[(4-fluorophenyl)methyl]piperazin-2-one
2-methyl-N-[1-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
5-[(3,4-dimethoxyphenyl)methyl]-5-{3-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
9-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-6-(pyridin-4-yl)-N-[3-(pyrrolidin-1-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[2-(3-chlorophenyl)ethyl]-1-{2-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-3-hydroxypropan-1-one
(4aS,7aR)-1-[(2-ethylphenyl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4-methoxy-2-methylphenyl)methyl]-N-(pyridin-3-ylmethyl)cyclopropanamine
1-[4-(4-ethyl-5-methylthiophene-3-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
(3S,7S)-5-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-N-(2-methylpropyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(3,4-dimethoxyphenyl)propyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
4-[4-(dimethylamino)benzoyl]-6-methoxy-1-[(4-methoxyphenyl)methyl]-1,4-diazepan-2-one
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(trifluoromethyl)benzamide
3-({6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3-diazinane-2,4-dione
2-{2-[(3,5-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}acetic acid
5-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-1H-1,2,4-triazol-3-amine
3-(5-methylfuran-2-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide