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N-benzyl-N-butyl-3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-(1-{1-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}ethyl)morpholine
2-(dimethyl-1,3-thiazol-2-yl)-7-ethyl-2,7-diazaspiro[4.5]decan-6-one
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-5-butyl-6-methyl-3,4-dihydropyrimidin-4-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1H-indol-2-ylmethyl)(methyl)[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amine
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}acetamide
5-cyclopropyl-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1,2-oxazole-4-carboxamide
4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-N-(2-ethoxyethyl)benzene-1-sulfonamide
(4aS,8aR)-1-(3-methylbutyl)-6-[2-(pyrimidin-2-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-[(5-{1-[(2-ethylphenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
N,N-diethyl-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-(4-methanesulfonylphenyl)-3-methyl-3-[(1-phenylpyrrolidin-3-yl)methyl]urea
1-[(2,6-dichloro-3-hydroxyphenyl)methyl]azepan-4-ol
5-benzyl-5-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
[4-(2-phenylethyl)-1-(pyridine-4-carbonyl)piperidin-4-yl]methanol
N-cyclopropyl-3-[1-(2-phenoxypropanoyl)piperidin-4-yl]propanamide
{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}[3-(methylsulfanyl)propyl]amine
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidine
4-[2-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-2-yl)ethyl]phenol
(4aR,8aS)-1-(2-cyclohexylethyl)-6-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
3-[1-(oxan-4-yl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
(3S,4S)-4-(4-fluorophenyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidin-3-ol
2-(dimethylamino)-N-(3-methyl-1-{7-[4-(2-methylpropyl)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
2-methanesulfonamido-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
3-{[(1R,5S,8S)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]sulfonyl}-N-[3-(methylsulfanyl)propyl]benzamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-fluorobenzamide
5-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrazin-2-amine
6-(3-chlorobenzoyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
3-(2-amino-1,3-thiazol-4-yl)-1-{3-[4-(hydroxymethyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
7-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-ethyl-N-[2-(3-methoxyphenoxy)ethyl]isoquinoline-3-carboxamide
N-methyl-N-[3-(morpholin-4-yl)propyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-{4-[(cyclopent-3-en-1-yl)amino]-2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
6-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
3-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}benzoic acid
6-[(diethylamino)methyl]-N-[(1S,2S)-2-hydroxycyclohexyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]butan-1-one
4-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
N-(4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}phenyl)acetamide
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]acetamide
3-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)propan-1-ol
N-[3-(1H-imidazol-1-yl)propyl]-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
(3R,4R)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine-2-carbonitrile
1-[(3-acetylphenyl)methyl]-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
3-(2-methoxyethyl)-1-(1-methyl-1H-pyrazol-4-yl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea