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8-{[4-(2-hydroxyethoxy)phenyl]methyl}-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(pyridin-3-yl)-1-{[4-(quinoxalin-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-4-ol
5-(4-chloro-2-methoxyphenoxymethyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
4-[3-(pyrrolidin-1-yl)propyl]-N-(quinolin-6-yl)-1,4-diazepane-1-carboxamide
methyl 3-benzamido-5-{[(3-methylphenyl)formamido]methyl}benzoate
N-{[1-(2-methoxyethyl)piperidin-3-yl]methyl}-N-methyl-4-(5-methylfuran-2-yl)benzamide
(5-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
4-[6-(benzyloxy)-4-cyclohexyl-3-oxo-1,4-diazepan-1-yl]-4-oxobutanamide
2-[(3,5-difluorophenyl)methyl]-8-(2-methylfuran-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
5-(2-methoxyphenoxymethyl)-N-{spiro[2.5]octan-1-ylmethyl}-1,2-oxazole-3-carboxamide
3-(1-{1-[2-(4-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
6-methyl-N-[(2-methyl-1H-imidazol-4-yl)methyl]-2H-1,3-benzodioxol-5-amine
4-[1-(2,3-dihydro-1H-inden-2-yl)-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-3-yl]pyridine
dimethyl({2-[4-(2-methylquinoline-4-carbonyl)morpholin-2-yl]ethyl})amine
2-[1-(propan-2-yl)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl]ethan-1-ol
1-[(3-fluorophenyl)methyl]-4-{imidazo[1,2-b]pyridazine-3-carbonyl}piperazine
2-[hydroxy(phenyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
5-methyl-5-phenyl-1-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-2-one
8-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-2,1,3-benzoxadiazole
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
1-cyclopentyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
N-[(3-chlorophenyl)methyl]-1-cyclopropyl-N-methyl-6-oxopiperidine-3-carboxamide
1-[2-(dimethylamino)ethyl]-6-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-oxo-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
8-[(2-hydroxy-5-methoxyphenyl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-[(2-fluorophenyl)methyl]-2-[1-(2-phenylethyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1-cyclopropyl-1H-pyrrole-2-carboxamide
1-{2-[6-hydroxy-4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,4-diazepan-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
7-[(4-fluorophenyl)methyl]-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
8-[(5-acetylthiophen-3-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-4-({3-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]-1H-pyrazol-1-yl}methyl)-1,3-thiazole
methyl 3-(3,4-dimethylbenzoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-phenyl-N-[2-(1,3-thiazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-methyl-3-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-2-yl)-1,2-oxazole
1,3-dimethyl-6-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,3-oxazole-4-carboxamide
2-methoxy-N-[(2R,3R)-2-methoxy-1'-[(3-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
3-(2-methylpropyl)-5-({4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}methyl)-1,2-oxazole
methyl[(3-{2-[4-(4-methylbenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
3-({4-methyl-6-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]pyrimidin-2-yl}amino)phenol
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(thiophen-2-ylmethyl)propanamide
2-[5-cyclopropyl-4-(piperidine-1-carbonyl)-1H-pyrazol-1-yl]-4-(3-fluoro-4-methoxyphenyl)pyrimidine
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
1-{3-[3-(4-ethylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propyl}-3,5-dimethyl-1H-pyrazole
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)urea
ethyl 4-{[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
1-[1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)azetidin-3-yl]-2-methylpiperidine
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(6-methylpyridin-2-yl)methyl]acetamide